Proteases
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GI 254023X
Catalog No. A15322 ADAM10 metalloprotease 抑制剂GI 254023X是一种选择性的ADAM10金属蛋白酶抑制剂;与ADAM17相比,ADAM10的效能高出100倍以上。 了解更多 -
Elastase Inhibitor, SPCK
Catalog No. A14913 -
Carboxypeptidase G2 (CPG2) Inhibitor
Catalog No. A15035 -
ZJ 43
Catalog No. A15318 -
Aloin (Barbaloin)
Catalog No. A10058 -
Arbutin (Uva, p-Arbutin)
Catalog No. A10084 Tyrosinase 抑制剂Arbutin (Uva,p-Arbutin)是用于中药(TCM)的糖基化对苯二酚。 熊果苷由于其酪氨酸酶抑制活性而抑制黑色素的形成。 了解更多 -
4-Chlorophenylguanidine hydrochloride
Catalog No. A15324 -
BC 11 hydrobromide
Catalog No. A15325 Urokinase (uPA) 抑制剂BC 11 hydrobromide是一种选择性尿激酶(uPA)抑制剂(IC50 = 8.2μM)。抑制血块溶解,不影响血块形成,对其他8种与uPA相关的酶也没有活性。 了解更多 -
GGACK Dihydrochloride
Catalog No. A16057 Urokinase 抑制剂GGACK Dihydrochloride是尿激酶(uPA(ICkin <1 ?M),凝血因子VIIa,凝血因子IXa,凝血因子Xa和胰蛋白酶的有效且不可逆的抑制剂。 了解更多 -
CTS-1027
Catalog No. A11345 -
Batimastat (BB-94)
Catalog No. A12985 MMP 抑制剂Batimastat (BB-94)是多种基质金属蛋白酶(MMP)的强效合成抑制剂,包括间质胶原酶(IC50 = 3 nM),溶血素(IC50 = 20 nM),Mr 72,000型IV胶原酶(IC50 = 4) nM),92,000型IV胶原酶先生(IC50 = 4 nM)和基质溶素(IC50 = 6 nM)。它是一种低分子量(MW = 478)的肽样胶原蛋白底物类似物,由类似物结合而成,分别与MMP和催化活性锌原子结合在一起。 了解更多 -
TAPI-0
Catalog No. A13724 -
Abametapir
Catalog No. A15945 metalloproteinase 抑制剂ABAMETAPIR是Xeglyze乳液的活性成分。ABAMETAPIR抑制金属蛋白酶;对卵子发育,若虫和成年虱子存活至关重要的生理过程必不可少的酶。 了解更多 -
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最新产品
Incyclinide
Catalog No. A17240 MMP inhibitorIincyclinide, also known as CMT-3 and COL-3, is a MMP inhibitor and a chemically-modified tetracycline with potential antineoplastic activity. Incyclinide inhibits matrix metalloproteinases (MMPs), thereby inducing extracellular matrix degradation, and inhibiting angiogenesis, tumor growth and invasion, and metastasis. This agent also causes mitochondrial depolarization in tumor cells and induces both cellular apoptosis and tissue necrosis. 了解更多 -
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4-epi-Chlortetracycline Hydrochloride
Catalog No. A12848 MMP 抑制剂4-epi-Chlortetracycline Hydrochloride是一种四环素衍生物,可作为金属蛋白酶(MMP)抑制剂,用于治疗组织破坏性疾病和癌症。 了解更多 -
NSC 405020
Catalog No. A13072 MT1-MMP 抑制剂NSC-405020是一种膜1型基质金属蛋白酶(MT1-MMP)抑制剂(IC50> 100μmol/ L)。 了解更多 -
Marimastat
Catalog No. A12826 -
GM 6001
Catalog No. A13320 -
SB-3CT
Catalog No. A14253 -
CL-82198
Catalog No. A13597 -
ARP 101
Catalog No. A15293 -
UK 370106
Catalog No. A15316 -
Batimastat sodium salt
Catalog No. A15326 MMP 抑制剂Batimastat sodium salt是一种抗癌药物,属于称为血管生成抑制剂的药物家族。Batimastat(BB-94)是一种有效的广谱基质金属蛋白酶(MMP)抑制剂。 了解更多 -
20(R)-Ginsenoside Rh2
Catalog No. A15408 -
Doxycycline
Catalog No. A17545 MMP inhibitorDoxycycline, an antibiotic, is an orally active and broad-spectrum metalloproteinase (MMP) inhibitor. 了解更多 -
Doxycycline monohydrate
Catalog No. A17813 MMP inhibitorDoxycycline monohydrate is an antibiotic and broad-spectrum metalloproteinase (MMP) inhibitor. 了解更多 -
Apratastat
Catalog No. A13330 dual TACE/MMPs inhibitorApratastat is an orally active, potent, and reversible dual inhibitor of tumor necrosis factor-α converting enzyme (TACE) and matrix metalloproteinases (MMPs) . 了解更多 -
MMP3 inhibitor 1
Catalog No. A13185 MMP-3 inhibitorMMP3 inhibitor 1 is a potent and highly selective MMP-3 inhibitor with an IC50 of 1 nM. 了解更多 -
BIBR-1048 (Dabigatran etexilate)
Catalog No. A10139 Thrombin 抑制剂BIBR-1048 (Dabigatran etexilate)是dabigatran的前体药物,dabigatran是一种有效的、非肽类小分子化合物,可特异地、可逆性地抑制游离的和结合了血凝块的凝血酶。 了解更多 -
BIBR 953 (Dabigatran, Pradaxa)
Catalog No. A10138 Thrombin 抑制剂BIBR 953 (Dabigatran,Pradaxa)是一种高度选择性,可逆且有效的凝血酶抑制剂,可作为前药达比加群酯口服。它在血栓形成的动物模型中显示出抗血栓形成的功效,起效迅速,可预测的药效学反应。 了解更多 -
Argatroban
Catalog No. A11774