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BIBR-1048 (Dabigatran etexilate)
Catalog No. A10139 Thrombin 抑制剂BIBR-1048 (Dabigatran etexilate)是dabigatran的前体药物，dabigatran是一种有效的、非肽类小分子化合物，可特异地、可逆性地抑制游离的和结合了血凝块的凝血酶。 了解更多 -
BIBR 953 (Dabigatran, Pradaxa)
Catalog No. A10138 Thrombin 抑制剂BIBR 953 (Dabigatran,Pradaxa)是一种高度选择性，可逆且有效的凝血酶抑制剂，可作为前药达比加群酯口服。它在血栓形成的动物模型中显示出抗血栓形成的功效，起效迅速，可预测的药效学反应。 了解更多 -
Argatroban
Catalog No. A11774 -
Bivalirudin
Catalog No. A15023 -
Dabigatran etexilate mesylate
Catalog No. A15057 direct thrombin 抑制剂Dabigatran etexilate mesylate是达比加群的口服活性前药。达比加群是一种可逆的选择性直接凝血酶抑制剂（DTI），Ki值为4.5 nM。 了解更多 -
Dabigatran ethyl ester
Catalog No. A15058 -
Eltrombopag Olamine
Catalog No. A15078 c-mpl (TpoR) receptor 激动剂Eltrombopag olamine是一种新型的口服活性血小板生成素受体（c-mpl）激动剂，可刺激血小板生成。 了解更多 -
Avatrombopag
Catalog No. A14087 -
Ximelagatran
Catalog No. A12509 -
TPO agonist 1
Catalog No. A16287 -
Melagatran
Catalog No. A19083 Thrombin inhibitorMelagatran is a direct and orally active inhibitor of thrombin, without interacting with any other enzymes in the coagulation cascade or fibrinolytic enzymes aside from thrombin. 了解更多 -
RWJ-445167
Catalog No. A12154 dual inhibitor of thrombin and factor XaRWJ-445167 (3DP-10017) is a dual inhibitor of thrombin and factor Xa with Ki of 4.0 nM and 230 nM, respectively, exhibiting potent antithrombotic activity. 了解更多 -
Thrombin Inhibitor 2
Catalog No. A21814 thrombin inhibitorThrombin Inhibitor 2 is a small molecule direct thrombin inhibitor, extracted from US8541580B2. Thrombin Inhibitor 2 has antithrombotic activity. 了解更多 -
CHR2797 (Tosedostat)
Catalog No. A10208 Aminopeptidase 抑制剂CHR2797 (Tosedostat)是一种新型金属酶抑制剂，在体内和体外对多种肿瘤细胞系均具有抗增殖作用，并表现出选择性。 了解更多 -
Bestatin Methyl Ester
Catalog No. A13592 Aminopeptidase 抑制剂Bestatin Methyl Ester是Bestatin的细胞可渗透衍生物，其对中性氨肽酶的抑制比Bestatin稍强，但对碱性氨肽酶的活性弱得多。 了解更多 -
Fumagillin
Catalog No. A15299 Aminopeptidase 抑制剂Fumagillin是一种复杂的天然产物抗生素，它与II型蛋氨酸氨基肽酶（MetAP-2）的关键组氨酸残基共价结合，抑制内皮细胞增殖和血管生成。 了解更多 -
Nafamostat mesylate
Catalog No. A10617 serine protease 抑制剂Nafamostat mesylate是一种抗凝剂。广谱丝氨酸蛋白酶抑制剂。在哮喘小鼠模型中减少嗜酸性粒细胞浸润，肥大细胞活化和气道反应性。 了解更多 -
BCX 1470
Catalog No. A11331 -
BCX 1470 methanesulfonate
Catalog No. A11325 Serine protease 抑制剂BCX 1470 methanesulfonate是丝氨酸蛋白酶抑制剂。BCX 1470在体外阻断补体酶CLs和因子D的酯酶和溶血活性。 了解更多 -
Camostat mesylate
Catalog No. A11764 Camostat mesylate是胰蛋白酶样的蛋白酶抑制剂，抑制胰蛋白酶和各种炎症性蛋白酶，包括纤溶酶，激肽释放酶和凝血酶。 了解更多 -
Sivelestat sodium salt
Catalog No. A14073 Neutrophil elastase 抑制剂Sivelestat sodium salt是一种选择性白细胞弹性蛋白酶抑制剂（IC50 = 44 nM），在一系列其他蛋白酶中均无活性。它在体外抑制NF-κB活化和LTB4诱导的中性粒细胞转运。 了解更多 -
Alvelestat
Catalog No. A12779 neutrophil elastase 抑制剂Avelestat，也称为AZD9668，是可口服的,高度选择性neutrophil elastase (NE)抑制剂，IC50和Ki分别为12 nM和9.4 nM,其选择性超过其他丝氨酸蛋白酶至少600倍。 了解更多 -
AEBSF HCl
Catalog No. A14270 -
Sivelestat
Catalog No. A14184 Neutrophil elastase 抑制剂Sivelestat是一种可渗透细胞的磺酰苯胺化合物，可作为中性粒细胞弹性蛋白酶的强效，底物竞争性和高度特异性抑制剂（大鼠，兔，仓鼠，人类和小鼠白细胞弹性蛋白酶的IC50 = 19-49 nM）。 了解更多 -
SSR 69071
Catalog No. A15315 -
PMSF
Catalog No. A11901 -
Sivelestat sodium hydrate (ONO-5046 sodium hydrate)
Catalog No. A16137 Neutrophil elastase 抑制剂Sivelestat sodium hydrate (ONO-5046 sodium hydrate)是人嗜中性粒细胞弹性蛋白酶的竞争性抑制剂，还抑制从兔，大鼠，仓鼠和小鼠获得的白细胞弹性蛋白酶。 了解更多 -
Fumonisin B1
Catalog No. A15379 serine/threonine phosphatase 抑制剂Fumonisin B1是由镰孢镰刀菌（Fusarium moniliforme）产生的真菌代谢产物，已显示可抑制蛋白质丝氨酸/苏氨酸磷酸酶（PP1，PP2A，PP2B，PP2C和PP5/T/K/H），并且对PP5最有效。 了解更多 -
Nafamostat hydrochloride
Catalog No. A20828 serine protease inhibitorNafamostat hydrochloride is an anticoagulant. Broad spectrum serine protease inhibitor. Reduces eosinophil infiltration, mast cell activation and airway responsiveness in a murine model of asthma. 了解更多 -
Nafamostat
Catalog No. A20827 serine protease inhibitorNafamostat is an anticoagulant. Broad spectrum serine protease inhibitor. Reduces eosinophil infiltration, mast cell activation and airway responsiveness in a murine model of asthma. 了解更多 -
Odanacatib (MK-0822)
Catalog No. A11265 -
CA-074
Catalog No. A13256 -
E 64d (Aloxistatin)
Catalog No. A13259 Cysteine Protease 抑制剂E 64d (Aloxistatin)是组织蛋白酶B和L的抑制剂，具有溶酶体和细胞渗透性。 了解更多 -
Leupeptin hemisulfate
Catalog No. A14145 -
Loxistatin Acid (E64-C)
Catalog No. A13258 -
E-64
Catalog No. A13257 -
Gly-Phe-beta-naphthylamide
Catalog No. A13611 cathepsin C substrateGly-Phe-beta-naphthylamide-萘酰胺是组织蛋白酶c底物。该化合物被描述为积聚在溶酶体内部，导致溶酶体的破坏。 了解更多 -
CA-074 Methyl Ester
Catalog No. A13593 Cathepsin B 抑制剂CA-074 Methyl Ester是CA-074的细胞渗透性类似物，用作不可逆组织蛋白酶B抑制剂。据报道，CA-074甲酯在啮齿动物模型中抑制骨吸收，并显示在体外抑制B16黑素瘤细胞侵袭。 了解更多 -
Z-FL-COCHO
Catalog No. A13502 -
SID 26681509
Catalog No. A15313
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