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RG2833 (RGFP109)

RG2833 (RGFP109)

Name: RG2833 (RGFP109)
SKU: A13139

目录号: A13139

HDAC 抑制剂

RG2833 (RGFP109) Chemical Structure

CAS NO. 1215493-56-3

RG2833 (RGFP109)是一种脑渗透性HDAC抑制剂，IC50为60 nM，HDAC1和HDAC3为50 nM。

库存：现货

规格	价格	数量
10 mg	￥ 490.00
25 mg	￥ 910.00
50 mg	￥ 1,330.00
10mM * 1mL in DMSO	￥ 602.00

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生物活性

RG2833 (RGFP109)是一种脑渗透性HDAC抑制剂，IC50为60 nM，HDAC1和HDAC3为50 nM。

靶点信息

HDAC3 (Cell-free assay)	HDAC1 (Cell-free assay)	HDAC3 (Cell-free assay)	HDAC1 (Cell-free assay)
5 nM(Ki)	32 nM(Ki)	5 nM(Ki)	32 nM(Ki)

溶解度 *

In vitro	DMSO	65 mg/mL (191.49 mM)
	Water	Insoluble
	Ethanol	10 mg/mL (29.46 mM)
* <1 mg/ml means slightly soluble or insoluble. * Please note that Adooq tests the solubility of all compounds in-house, and the actual solubility may differ slightly from published values. This is normal and is due to slight batch-to-batch variations.

制备储备液

Concentration / Solvent Volume / Mass	1 mg	5 mg	10 mg
0.1 mM	29.46 mL	147.31 mL	294.61 mL
0.5 mM	5.89 mL	29.46 mL	58.92 mL
1 mM	2.95 mL	14.73 mL	29.46 mL
5 mM	0.59 mL	2.95 mL	5.89 mL

*The above data is based on the productmolecular weight 339.43. Batch specific molecular weights may vary from batch to batch due to solvent of hydration, which will affect the solvent volumes required to prepare stock solutions.

化学数据

目录号	A13139
作用机制	Inhibitor (抑制剂)
M. Wt	339.43
Formula	C20H25N3O2
Purity	>99%
Storage	Store lyophilized at -20ºC, keep desiccated. In lyophilized form, the chemical is stable for 36 months. In solution, store at -20ºC and use within 3 months to prevent loss of potency. Aliquot to avoid multiple freeze/thaw cycles.
CAS No.	1215493-56-3
Synonyms	RGFP109
SMILES	CC1=CC=C(C=C1)C(=O)NCCCCCC(=O)NC2=CC=CC=C2N