你的浏览器似乎禁用了 JavaScript。
您必须在浏览器中启用JavaScript才能使用本网站的功能。

微信关注
申请试用装

主页 /
Membrane Transporters/Ion Channels /
Sodium Channels

Sodium Channels

Quick View
Raxatrigine hydrochloride

Catalog No. A21645
Quick View

添加到收藏
Nav1.7 sodium channel inhibitor

Raxatrigine hydrochloride (GSK-1014802 hydrochloride) is a novel small molecule state-dependent sodium channel blocker; Nav1.7 sodium channel inhibitor. 了解更多

Bulk Inquiry
Quick View
Funapide

Catalog No. A21298
Quick View

添加到收藏
Sodium Channel Nav1.7 inhibitor

Funapide (TV 45070; XEN402) is a potent Sodium Channel Nav1.7 inhibitor. 了解更多

Bulk Inquiry
Quick View
Nav1.7-IN-3

Catalog No. A13626
Quick View

添加到收藏
voltage-gated sodium channel Nav1.7 inhibitor

Nav1.7-IN-3 is a selective, orally bioavailable voltage-gated sodium channel Nav1.7 inhibitor with an IC50 of 8 nM. Pain relief. Limited CNS penetration. 了解更多

Bulk Inquiry
Quick View
ICA-121431

Catalog No. A13773
Quick View

添加到收藏
NaV1.3 and NaV1.1 channels 抑制剂

ICA-121431是人NaV1.3和NaV1.1通道的有效和选择性抑制剂（IC50值分别为13和23 nM）。了解更多

Bulk Inquiry Free Sample
Quick View
S0859

Catalog No. A15228
Quick View

添加到收藏
NBC 抑制剂

S0859是一种N-氰基磺酰胺化合物，可逆地抑制NBC介导的pH（i）恢复（K（i）= 1.7 microM，在约30 microM处完全抑制）。了解更多

Bulk Inquiry Free Sample
Quick View
Sodium Channel inhibitor 1

Catalog No. A15243
Quick View

添加到收藏
Sodium Channel 抑制剂

Sodium Channel inhibitor 1 是一种新型的选择性电压门控钠通道，用于疼痛治疗。了解更多

Bulk Inquiry
Quick View
GS967

Catalog No. A14361
Quick View

添加到收藏
late INa 抑制剂

GS967是一种新型的，有效的，选择性的心脏晚期钠电流抑制剂（INa晚期）；抑制心室肌细胞和离体心脏中ATX-II诱导的晚期I（Na），IC（50）值分别为0.13和0.21 uM。了解更多

Bulk Inquiry
Quick View
Levobupivacaine

Catalog No. A15979
Quick View

添加到收藏
sodium channel 抑制剂

Levobupivacaine是属于氨基酰胺类的局部麻醉药。了解更多

Bulk Inquiry
Quick View
Procaine

Catalog No. A16131
Quick View

添加到收藏
voltage-gated sodium channel 抑制剂

Procaine是具有局麻和抗心律不齐特性的苯甲酸衍生物。了解更多

Bulk Inquiry
Quick View
PF-05089771

Catalog No. A16365
Quick View

添加到收藏
Nav1.7 抑制剂

PF-05089771是一种选择性Nav1.7抑制剂（IC50 = 11 nM），与域IV的电压传感器域（VSD）相互作用。了解更多

Bulk Inquiry
Quick View
Ambroxol HCl

Catalog No. A16398
Quick View

添加到收藏
Sodium Channel 抑制剂

Ambroxol HCl是神经元Na+通道的有效抑制剂，可抑制TTX耐受的Na+电流，IC50为35.2 uM，对于补品和相阻滞的IC50为22.5 μM，抑制TTX敏感的Na+电流，IC50为100 μM。第三阶段。了解更多

Product Citations (1)

Bulk Inquiry
- Giovanni Bocci, .et al. Virtual and In Vitro Antiviral Screening Revive Therapeutic Drugs for COVID-19, ACS Pharmacol Transl Sci, 2020, Oct 14
Quick View
PF-04971729

Catalog No. A11102
Quick View

添加到收藏
SGLT2 抑制剂

PF-04971729是钠依赖性葡萄糖共转运蛋白2的有效和选择性抑制剂。了解更多

Bulk Inquiry
Quick View
Orphenadrine citrate

Catalog No. A11712
Quick View

添加到收藏
NMDA receptor 拮抗剂

Orphenadrine柠檬酸盐是NMDA受体拮抗剂，Ki为6.0μM，还是HERG钾离子通道阻断剂。了解更多

Bulk Inquiry Free Sample
Quick View
Vinpocetine

Catalog No. A11602
Quick View

添加到收藏
PDE1 抑制剂

Vinpocetine是一种Ca2+钙调蛋白依赖性磷酸二酯酶I（PDE1）抑制剂。了解更多

Bulk Inquiry
Quick View
ENIPORIDE

Catalog No. A14139
Quick View

添加到收藏
Na(+)/H(+) exchange 抑制剂

ENIPORIDE是一种有效的Na+/H+交换抑制剂。了解更多

Bulk Inquiry
Quick View
Digoxin

Catalog No. A14242
Quick View

添加到收藏
sodium-potassium pump 抑制剂

Digoxin是Na+/K+-ATPase 的有效抑制剂了解更多

Product Citations (1)

Bulk Inquiry Free Sample
- Reiko Watanabe, .et al. Development of an In Silico Prediction Model for P-glycoprotein Efflux Potential in Brain Capillary Endothelial Cells toward the Prediction of Brain Penetration, J Med Chem, 2021, Mar 11;64(5):2725-2738 PMID: 33619967
Quick View
Procainamide HCl

Catalog No. A14240
Quick View

添加到收藏
Sodium channel blocker/DNMT 抑制剂

Procainamide HCl是钠通道阻滞剂，又是DNA甲基转移酶抑制剂。了解更多

Bulk Inquiry
Quick View
Oxcarbazepine

Catalog No. A13943
Quick View

添加到收藏
sodium channel protein 抑制剂

Oxcarbazepine是一种钠通道蛋白抑制剂。了解更多

Bulk Inquiry

溶液配制计算器

分子量计算器

稀释计算器

摩尔浓度计算器

ADOOQ 产品质量保证

Guaranteed product quality, 365 days Unconditional Return & Replacement

We promise all products to perform as described.