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Membrane Transporters/Ion Channels /
Sodium Channels

Sodium Channels

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Raxatrigine hydrochloride

Catalog No. A21645
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Nav1.7 sodium channel inhibitor

Raxatrigine hydrochloride (GSK-1014802 hydrochloride) is a novel small molecule state-dependent sodium channel blocker; Nav1.7 sodium channel inhibitor. 了解更多

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Funapide

Catalog No. A21298
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Sodium Channel Nav1.7 inhibitor

Funapide (TV 45070; XEN402) is a potent Sodium Channel Nav1.7 inhibitor. 了解更多

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Nav1.7-IN-3

Catalog No. A13626
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voltage-gated sodium channel Nav1.7 inhibitor

Nav1.7-IN-3 is a selective, orally bioavailable voltage-gated sodium channel Nav1.7 inhibitor with an IC50 of 8 nM. Pain relief. Limited CNS penetration. 了解更多

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ICA-121431

Catalog No. A13773
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NaV1.3 and NaV1.1 channels 抑制剂

ICA-121431是人NaV1.3和NaV1.1通道的有效和选择性抑制剂（IC50值分别为13和23 nM）。了解更多

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S0859

Catalog No. A15228
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NBC 抑制剂

S0859是一种N-氰基磺酰胺化合物，可逆地抑制NBC介导的pH（i）恢复（K（i）= 1.7 microM，在约30 microM处完全抑制）。了解更多

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Sodium Channel inhibitor 1

Catalog No. A15243
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Sodium Channel 抑制剂

Sodium Channel inhibitor 1 是一种新型的选择性电压门控钠通道，用于疼痛治疗。了解更多

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GS967

Catalog No. A14361
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late INa 抑制剂

GS967是一种新型的，有效的，选择性的心脏晚期钠电流抑制剂（INa晚期）；抑制心室肌细胞和离体心脏中ATX-II诱导的晚期I（Na），IC（50）值分别为0.13和0.21 uM。了解更多

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Levobupivacaine

Catalog No. A15979
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sodium channel 抑制剂

Levobupivacaine是属于氨基酰胺类的局部麻醉药。了解更多

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Procaine

Catalog No. A16131
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voltage-gated sodium channel 抑制剂

Procaine是具有局麻和抗心律不齐特性的苯甲酸衍生物。了解更多

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PF-05089771

Catalog No. A16365
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Nav1.7 抑制剂

PF-05089771是一种选择性Nav1.7抑制剂（IC50 = 11 nM），与域IV的电压传感器域（VSD）相互作用。了解更多

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Ambroxol HCl

Catalog No. A16398
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Sodium Channel 抑制剂

Ambroxol HCl是神经元Na+通道的有效抑制剂，可抑制TTX耐受的Na+电流，IC50为35.2 uM，对于补品和相阻滞的IC50为22.5 μM，抑制TTX敏感的Na+电流，IC50为100 μM。第三阶段。了解更多

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- Giovanni Bocci, .et al. Virtual and In Vitro Antiviral Screening Revive Therapeutic Drugs for COVID-19, ACS Pharmacol Transl Sci, 2020, Oct 14
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PF-04971729

Catalog No. A11102
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SGLT2 抑制剂

PF-04971729是钠依赖性葡萄糖共转运蛋白2的有效和选择性抑制剂。了解更多

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Orphenadrine citrate

Catalog No. A11712
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NMDA receptor 拮抗剂

Orphenadrine柠檬酸盐是NMDA受体拮抗剂，Ki为6.0μM，还是HERG钾离子通道阻断剂。了解更多

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Vinpocetine

Catalog No. A11602
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PDE1 抑制剂

Vinpocetine是一种Ca2+钙调蛋白依赖性磷酸二酯酶I（PDE1）抑制剂。了解更多

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ENIPORIDE

Catalog No. A14139
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Na(+)/H(+) exchange 抑制剂

ENIPORIDE是一种有效的Na+/H+交换抑制剂。了解更多

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Digoxin

Catalog No. A14242
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sodium-potassium pump 抑制剂

Digoxin是Na+/K+-ATPase 的有效抑制剂了解更多

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- Reiko Watanabe, .et al. Development of an In Silico Prediction Model for P-glycoprotein Efflux Potential in Brain Capillary Endothelial Cells toward the Prediction of Brain Penetration, J Med Chem, 2021, Mar 11;64(5):2725-2738 PMID: 33619967
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Procainamide HCl

Catalog No. A14240
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Sodium channel blocker/DNMT 抑制剂

Procainamide HCl是钠通道阻滞剂，又是DNA甲基转移酶抑制剂。了解更多

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Oxcarbazepine

Catalog No. A13943
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sodium channel protein 抑制剂

Oxcarbazepine是一种钠通道蛋白抑制剂。了解更多

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