SP2509 (HCI-2509)

Name: SP2509 (HCI-2509)
SKU: A14443

目录号: A14443

LSD1 抑制剂

SP2509 (HCI-2509) Chemical Structure

CAS NO. 1423715-09-6

SP2509 (HCI-2509)是一种新型组蛋白脱甲基酶LSD1（KDM1A）拮抗剂，IC50为13 nM。对MAO-A和MAO-B没有抑制作用。

库存：现货

规格	价格	数量
5 mg	￥ 385.00
10 mg	￥ 560.00
25 mg	￥ 1,155.00

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生物活性

SP2509 (HCI-2509)是一种新型组蛋白脱甲基酶LSD1（KDM1A）拮抗剂，IC50为13 nM。对MAO-A和MAO-B没有抑制作用。

靶点信息

LSD1
13 nM

溶解度 *

In vitro (25°C)	DMSO	36 mg/mL (82.2 mM)
	Water	Insoluble
	Ethanol	Insoluble
In vivo	10% DMSO+corn oil	4 mg/mL
* <1 mg/ml means slightly soluble or insoluble. * Please note that Adooq tests the solubility of all compounds in-house, and the actual solubility may differ slightly from published values. This is normal and is due to slight batch-to-batch variations.

制备储备液

Concentration / Solvent Volume / Mass	1 mg	5 mg	10 mg
0.1 mM	22.84 mL	114.18 mL	228.36 mL
0.5 mM	4.57 mL	22.84 mL	45.67 mL
1 mM	2.28 mL	11.42 mL	22.84 mL
5 mM	0.46 mL	2.28 mL	4.57 mL

*The above data is based on the productmolecular weight 437.9. Batch specific molecular weights may vary from batch to batch due to solvent of hydration, which will affect the solvent volumes required to prepare stock solutions.

化学数据

目录号	A14443
作用机制	Inhibitor (抑制剂)
M. Wt	437.9
Formula	C19H20ClN3O5S
Purity	>99%
Storage	Store lyophilized at -20ºC, keep desiccated. In lyophilized form, the chemical is stable for 36 months. In solution, store at -20ºC and use within 3 months to prevent loss of potency. Aliquot to avoid multiple freeze/thaw cycles.
CAS No.	1423715-09-6
Synonyms	SP-2509
SMILES	CC(=C1C=C(C=CC1=O)Cl)NNC(=O)C2=CC(=CC=C2)S(=O)(=O)N3CCOCC3