SR 144528

Name: SR 144528
SKU: A12376

目录号: A12376

CB2 inverse 激动剂

Product Citations (1)

SR 144528 Chemical Structure

CAS NO. 192703-06-3

SR 144528是一种选择性的外周大麻素受体反向激动剂，对大鼠脾脏和人重组CB2受体的Ki值为0.6 nM，对大鼠脑和人重组CB1受体的Ki值为400 nM。

库存：现货

规格	价格	数量
5 mg	￥ 665.00
10 mg	￥ 1,190.00
25 mg	￥ 2,730.00
50 mg	￥ 4,690.00

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生物活性

SR 144528是一种选择性的外周大麻素受体反向激动剂，对大鼠脾脏和人重组CB2受体的Ki值为0.6 nM，对大鼠脑和人重组CB1受体的Ki值为400 nM。

制备储备液

Concentration / Solvent Volume / Mass	1 mg	5 mg	10 mg
0.1 mM	21.01 mL	105.03 mL	210.06 mL
0.5 mM	4.2 mL	21.01 mL	42.01 mL
1 mM	2.1 mL	10.5 mL	21.01 mL
5 mM	0.42 mL	2.1 mL	4.2 mL

*The above data is based on the productmolecular weight 476.05. Batch specific molecular weights may vary from batch to batch due to solvent of hydration, which will affect the solvent volumes required to prepare stock solutions.

化学数据

目录号	A12376
作用机制	Agonist (激动剂)
M. Wt	476.05
Formula	C29H34ClN3O
Purity	>99%
Storage	Store lyophilized at -20ºC, keep desiccated. In lyophilized form, the chemical is stable for 36 months. In solution, store at -20ºC and use within 3 months to prevent loss of potency. Aliquot to avoid multiple freeze/thaw cycles.
CAS No.	192703-06-3
Synonyms	SR144528, SR-144528
SMILES	CC1=CC=C(C=C1)CN2C(=CC(=N2)C(=O)N[C@H]3[C@]4(CC[C@H](C4)C3(C)C)C)C5=CC(=C(C=C5)Cl)C