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TGR-1202 hydrochloride (Umbralisib HCl)

TGR-1202 hydrochloride (Umbralisib HCl)

Name: TGR-1202 hydrochloride (Umbralisib HCl)
SKU: A16278

目录号: A16278

PI3Kδ 抑制剂

TGR-1202 hydrochloride (Umbralisib HCl) Chemical Structure

CAS NO. 1532533-78-0

TGR-1202 hydrochloride是一种口服的下一代PI3Kδ抑制剂，在基于酶和细胞的测定中抑制PI3Kδ活性，IC50和EC50值分别为22.2和24.3 nM。

库存：现货

规格	价格	数量
5 mg	￥ 840.00
10 mg	￥ 1,540.00
50 mg	￥ 4,060.00

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生物活性

TGR-1202 hydrochloride是一种口服的下一代PI3Kδ抑制剂，在基于酶和细胞的测定中抑制PI3Kδ活性，IC50和EC50值分别为22.2和24.3 nM。

制备储备液

Concentration / Solvent Volume / Mass	1 mg	5 mg	10 mg
0.1 mM	16.45 mL	82.24 mL	164.47 mL
0.5 mM	3.29 mL	16.45 mL	32.89 mL
1 mM	1.64 mL	8.22 mL	16.45 mL
5 mM	0.33 mL	1.64 mL	3.29 mL

*The above data is based on the productmolecular weight 608.01. Batch specific molecular weights may vary from batch to batch due to solvent of hydration, which will affect the solvent volumes required to prepare stock solutions.

化学数据

目录号	A16278
作用机制	Inhibitor (抑制剂)
M. Wt	608.01
Formula	C31H25ClF3N5O3
Purity	>99%
Storage	Store lyophilized at -20ºC, keep desiccated. In lyophilized form, the chemical is stable for 36 months. In solution, store at -20ºC and use within 3 months to prevent loss of potency. Aliquot to avoid multiple freeze/thaw cycles.
CAS No.	1532533-78-0
Synonyms	RP5264 hydrochloride, TGR1202 hydrochloride, TGR 1202 hydrochloride, RP-5264 hydrochloride, RP 5264 hydrochloride
SMILES	O=C1C(C2=CC=CC(F)=C2)=C([C@@H](N3N=C(C4=CC=C(OC(C)C)C(F)=C4)C5=C(N)N=CN=C53)C)OC6=CC=C(F)C=C16.[H]Cl