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Membrane Transporters/Ion Channels

产品 201 到 250 共 317个

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  1. (S)-(-)-5-Fluorowillardiine
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    (S)-(-)-5-Fluorowillardiine

    Catalog No. A21337
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    AMPAR agonist
    (S)-(-)-5-Fluorowillardiine is a potent and specific AMPAR agonist. 了解更多
  2. Naspm trihydrochloride
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    Naspm trihydrochloride

    Catalog No. A21437
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    CP-AMPA receptors antagonist
    Naspm trihydrochloride (1-Naphthylacetyl spermine trihydrochloride), a synthetic analogue of Joro spider toxin, is a calcium permeable AMPA (CP-AMPA) receptors antagonist. 了解更多
  3. Fanapanel hydrate
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    Fanapanel hydrate

    Catalog No. A21668
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    AMPA/kainate antagonist
    Fanapanel hydrate (ZK200775 hydrate) is a highly selective AMPA/kainate antagonist with little activity against NMDA; have Ki values of 3.2 nM, 100 nM, and 8.5 μM against quisqualate, kainate, and NMDA, respectively. 了解更多
  4. Mibampator
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    Mibampator

    Catalog No. A21717
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    AMPA receptors potentiator
    Mibampator (LY451395) is a potent and highly selective potentiator of the AMPA receptors. 了解更多
  5. Philanthotoxin 74 dihydrochloride
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    Philanthotoxin 74 dihydrochloride

    Catalog No. A21739
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    AMPAR antagonist
    Philanthotoxin 74 dihydrochloride (PhTx 74) is an AMPAR antagonist; inhibits GluR3 and GluR1 with IC50s of 263 and 296 nM, respectively. 了解更多
  6. PEPA
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    PEPA

    Catalog No. A21904
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    AMPA receptors allosteric modulator
    PEPA is an allosteric modulator of AMPA receptors; binds to the GluA2o and GluA3o LBDs and can be utilized as an indicator of AMPA receptor heterogeneity. 了解更多
  7. CMPDA
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    CMPDA

    Catalog No. A21909
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    AMPA receptors positive allosteric modulator
    CMPDA is a positive allosteric modulator of AMPA receptors with EC50s of 45.4 ?? 4.2 nM/63.4 ?? 5.6 nM for GluA2i/GluA2o receptor. 了解更多
  8. Naspm
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    Naspm

    Catalog No. A21919
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    AMPA (CP-AMPA) receptors antagonist
    Naspm (1-Naphthyl acetyl spermine), a synthetic analogue of Joro spider toxin, is a calcium permeable AMPA (CP-AMPA) receptors antagonist. 了解更多
  9. Aniracetam
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    Aniracetam

    Catalog No. A10078
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    AMPA Receptor 抑制剂
    Aniracetam是一种安非他命，属于消旋体化学类别的促智药，据称比吡乙酰胺更有效。 了解更多
  10. Ampalex (CX-516)
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    Ampalex (CX-516)

    Catalog No. A12349
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    Ampalex (CX-516)是ampakine和nootropic，充当ampa受体阳性变构调节剂。 了解更多
  11. GYKI-52466 dihydrochloride
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    GYKI-52466 dihydrochloride

    Catalog No. A10444
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    AMPA and Kainate 拮抗剂
    GYKI-52466 dihydrochloride是选择性非竞争性AMPA受体拮抗剂(对于AMPA、红藻氨酸和AMPA诱导的反应，IC50值分别为10-20、~ 450和> > 50 μM)。 了解更多
  12. LY404187
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    LY404187

    Catalog No. A12424
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    LY404187是AMPA受体的选择性，有效和中枢活性的正构构调节剂。 了解更多
  13. LY450108
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    LY450108

    Catalog No. A12425
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    LY450108是一种α-氨基-3-羟基-5-甲基-4-异恶唑-丙酸（AMPA）受体增强剂。 了解更多
  14. NBQX
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    NBQX

    Catalog No. A13109
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    AMPA Receptor 拮抗剂
    NBQX是一种有效，选择性和竞争性的AMPA受体拮抗剂。 了解更多
  15. DNQX
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    DNQX

    Catalog No. A13882
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    NMDA receptor 拮抗剂
    DNQX是一种非N-甲基-D-天冬氨酸（非NMDA）受体复合物拮抗剂。 了解更多
  16. IEM 1754 Dihydrobromide
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    IEM 1754 Dihydrobromide

    Catalog No. A14010
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    AMPA Receptor Blocker
    IEM 1754 Dihydrobromide是AMPA受体的电压依赖性明渠阻断剂。 了解更多
  17. Farampator
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    Farampator

    Catalog No. A13798
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    AMPA receptor modulator
    Farampator是一种AMPA受体正调节剂，它可以改善短期记忆，但会损害情景记忆。 了解更多
  18. Cyclothiazide
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    Cyclothiazide

    Catalog No. A13700
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    AMPA desensitization 抑制剂
    Cyclothiazide是苯并噻二叠氮，可作为AMPA受体的增效剂，正向调节其对谷氨酸的响应（EC50 = 3.8 M）。 了解更多
  19. CNQX
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    CNQX

    Catalog No. A16109
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    AMPA/kainate 拮抗剂
    CNQX是一种竞争性的非NMDA谷氨酸受体拮抗剂（AMPA和海藻酸酯受体的IC50分别为0.3和1.5 uM，而NMDA受体的IC50 = 25 uM）。 了解更多
  20. CNQX disodium salt
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    CNQX disodium salt

    Catalog No. A16110
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    AMPA/kainate 拮抗剂
    CNQX disodium salt，AMPA/海藻酸酯拮抗剂CNQX（GLXC-11053）的水溶性形式。 了解更多
  21. GYKI53655 Hydrochloride
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    GYKI53655 Hydrochloride

    Catalog No. A17032
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    AMPA 拮抗剂
    GYKI53655 Hydrochloride是一种非竞争性AMPA和海藻酸酯受体拮抗剂。 了解更多
  22. CX546
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    CX546

    Catalog No. A21923
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    positive AMPAR modulator
    CX546 is a selective positive AMPAR modulator; the prototypical ampakine agent. 了解更多
  23. CFM-2
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    CFM-2

    Catalog No. A21930
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    non-competitive AMPAR antagonist
    CFM-2 is a selective non-competitive AMPAR antagonist. 了解更多
  24. (S)-Willardiine
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    (S)-Willardiine

    Catalog No. A21957
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    AMPA/kainate receptors agonist
    (S)-Willardiine is a potent agonist of AMPA/kainate receptors with EC50 of 44.8 uM. 了解更多
  25. Becampanel
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    Becampanel

    Catalog No. A21194
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    AMPA antagonist
    Becampanel (AMP397) is the first competitive AMPA antagonist and an antiepileptic agent. 了解更多
  26. Elacridar hydrochloride
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    Elacridar hydrochloride

    Catalog No. A15077
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    P-gp 抑制剂
    Elacridar hydrochloride是一种P-糖蛋白抑制剂，已在体内和体外用作P-糖蛋白（Pgp）的工具抑制剂，以研究转运蛋白在处理各种测试分子中的作用。 了解更多
  27. Zosuquidar
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    Zosuquidar

    Catalog No. A15289
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    P-gp 抑制剂
    Zosuquidar是P-糖蛋白介导的多药耐药性的有效调节剂，Ki为60 nM。 了解更多
  28. TTT-28
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    TTT-28

    Catalog No. A13033
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    ABCB1 (P-gp/MDR1) inhibitor
    TTT-28 is a synthesized thiazole-valine peptidomimetic, a novel selective inhibitor of ABCB1 (P-gp/MDR1) with high efficacy and low toxicity. 了解更多
  29. Norverapamil hydrochloride
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    Norverapamil hydrochloride

    Catalog No. A12249
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    P-gp inhibitor
    Norverapamil hydrochloride ((??)-Norverapamil hydrochloride), an N-demethylated metabolite of Verapamil, is a L-type calcium channel blocker and a P-glycoprotein (P-gp) function inhibitor. 了解更多
  30. P-gp inhibitor 1
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    P-gp inhibitor 1

    Catalog No. A13384
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    P-gp inhibitor
    P-gp inhibitor 1 is a novel inhibitor reversing P-glycoprotein-mediated multidrug resistance. 了解更多
  31. LY335979 (Zosuquidar 3HCl)
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    LY335979 (Zosuquidar 3HCl)

    Catalog No. A10549
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    P-gp modulator
    LY335979 (Zosuquidar trihydrochloride)是一种强效高选择性P-gp抑制剂。 了解更多
  32. PSC-833 (Valspodar)
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    PSC-833 (Valspodar)

    Catalog No. A11080
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    MDR1/P-gp 抑制剂
    PSC-833 (Valspodar)是一种P-糖蛋白（P-gp）调节剂，可抑制P-gp介导的多药耐药性（MDR）。 了解更多
  33. Elacridar (GF120918)
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    Elacridar (GF120918)

    Catalog No. A12324
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    P-gp & BCRP 抑制剂
    Elacridar (GF120918)是一种原型BCRP抑制剂，可抑制Bcrp1介导的转运。 了解更多
  34. Tariquidar (XR9576)
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    Tariquidar (XR9576)

    Catalog No. A11584
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    P-gp 抑制剂
    Tariquidar (XR9576)是一种P-糖蛋白药物外排泵抑制剂。 了解更多
  35. Selamectin
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    Selamectin

    Catalog No. A12363
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    Selamectin是一种局部寄生虫药和抗蠕虫药，用于狗和猫，以治疗和预防犬中的心丝虫，跳蚤，耳螨，螨和某些种类的壁虱感染，并预防心丝虫，跳蚤，耳螨，钩虫和round虫 在猫中。 了解更多
  36. Cynarin
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    Cynarin

    Catalog No. A12004
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    Cynarin是朝鲜蓟中的一种酚类化合物。它具有抗氧化剂和胆汁特性。它是一种潜在的免疫抑制剂。 了解更多
  37. XR9576
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    XR9576

    Catalog No. A13961
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    P-glycoprotein 抑制剂
    XR9576是一种 P-glycoprotein (P-gp) 抑制剂，Kd值为5.1 nM。正在研究中作为抗癌多药耐药性的佐剂。 了解更多
  38. ONT-093
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    ONT-093

    Catalog No. A13531
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    P-gp 抑制剂
    ONT-093是口服可生物利用的P-糖蛋白泵抑制剂，可潜在逆转接受癌症化学疗法的患者的多药耐药性。 了解更多
  39. Laniquidar
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    Laniquidar

    Catalog No. A13532
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    P-gp 抑制剂
    Laniquidar是第三代P-gp抑制剂，已在临床试验中用于调节多药耐药转运蛋白。 了解更多
  40. Biricodar dicitrate (VX-710 dicitrate)
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    Biricodar dicitrate (VX-710 dicitrate)

    Catalog No. A13533
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    P-gp modulator
    Biricodar dicitrate (VX-710 dicitrate)是P-糖蛋白和MRP-1的调节剂；在多药耐药细胞中显示出有效的化学增敏活性。 了解更多
  41. MC 70 HCl
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    MC 70 HCl

    Catalog No. A16080
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    P-gp 抑制剂
    MC 70 HCl是有效的P-gp抑制剂（EC50 = 0.69 uM）。 了解更多
  42. KS-176
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    KS-176

    Catalog No. A16195
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    BCRP 抑制剂
    KS-176是乳腺癌抗性蛋白（BCRP）多药转运蛋白的有效和选择性抑制剂（在Pheo A和Hoechst 33342分析中，IC50值分别为0.59和1.39 uM）。 了解更多
  43. FD 12-9
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    FD 12-9

    Catalog No. A18393
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    P-gp/BCRP dual 抑制剂
    FD 12-9 is a flavonoid dimer, acts as a dual inhibitor of P-gp and BCRP, with EC50s of 285 nM and 0.9 nM, respectively. Anti-glioblastoma activity. 了解更多
  44. Biricodar
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    Biricodar

    Catalog No. A21464
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    P-glycoprotein/MRP-1 modulator
    Biricodar (VX-710) is a modulator of P-glycoprotein and MRP-1; shows effective chemosensitizing activity in multidrug resistant cells. 了解更多
  45. Piperlongumine
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    Piperlongumine

    Catalog No. A14124
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    TrxR1/CRM1 抑制剂
    Piperlongumine，存在于胡椒科植物荜茇中的一种天然生物碱，能够增加reactive oxygen species (ROS)水平，并选择性杀死癌细胞。它还是TrxR1的直接抑制剂，对胃癌具有抑制活性；一种新型的CRM1抑制剂；在人类乳腺癌细胞中可抑制PI3K/Akt/mTOR。 了解更多
  46. KPT276
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    KPT276

    Catalog No. A16341
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    SINE/CRM1 抑制剂
    KPT276是KPT-185的类似物，是核出口（SINE）和CRM1的选择性抑制剂。 了解更多
  47. Eltanexor Z-isomer
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    Eltanexor Z-isomer

    Catalog No. A21786
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    CRM1 inhibitor
    Eltanexor Z-isomer (KPT-8602 Z-isomer) is the less active isomer of KPT-8602. KPT-8602 is a potent CRM1 inhibitor. 了解更多
  48. Leptomycin B
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    Leptomycin B

    Catalog No. A20985
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    nuclear export receptor CRM1 inhibitor
    Leptomycin B (CI 940; LMB) is a potent inhibitor of the nuclear export of proteins. Leptomycin B inactivates CRM1/exportin 1 by covalent modification at a cysteine residue. Leptomycin B is a potent antifungal antibiotic blocking the eukaryotic cell cycle. 了解更多
  49. KPT185
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    KPT185

    Catalog No. A12975
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    CRM1 抑制剂
    KPT185是选择性CRM1抑制剂。KPT-185以100 nM至500 nM的IC50显着抑制白血病细胞增殖，并诱导AML细胞系和原发性AML原始细胞的细胞周期停滞和凋亡。 了解更多
  50. Selinexor (KPT-330)
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    Selinexor (KPT-330)

    Catalog No. A12582
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    CRM1 抑制剂
    CRM1（XPO1）介导的核输出的KPT-330抑制剂在T细胞急性淋巴细胞白血病和急性骨髓性白血病的临床前模型中具有选择性的抗白血病活性。 了解更多

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购物选项

分类
  1. ATPase (22)
  2. CFTR (16)
  3. Calcium Channels (47)
  4. Sodium Channels (44)
  5. Potassium Channels (38)
  6. Chloride Channels (7)
  7. SGLT (15)
  8. Monocarboxylate transporters (MCT) (8)
  9. AMPA receptor (33)
  10. P-gp (19)
  11. CRM1 (6)
  12. TRP Channel (23)
  13. TRPV (15)
  14. Glutamate (EAAT) Transporters (1)
  15. Serotonin Transporter (3)
  16. Proton Pump (7)
  17. OCT (4)
  18. NCX (5)
  19. BCRP (6)
  20. MRP (1)
  21. Na+/H+ Exchanger (4)
  22. Monoamine Transporter (3)
作用机制
  1. Inhibitor (抑制剂) (122)
  2. Agonist (激动剂) (12)
  3. Antagonist (拮抗剂) (36)
  4. Activator (激活剂) (22)
  5. Modulator (调节剂) (15)
  6. Blocker (阻断剂) (47)
  7. Inducer (诱导剂) (3)
  8. Potentiator (增强剂) (5)
靶点
  1. DNMT (1)
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