YM201636

Name: YM201636
SKU: A11064

目录号: A11064

PI3K 抑制剂

Product Citations (2)

YM201636 Chemical Structure

CAS NO. 371942-69-7

YM201636是PIKfyve的细胞渗透性和选择性抑制剂（IC50 = 33 nM）。

库存：现货

规格	价格	数量
5 mg	￥ 630.00
10 mg	￥ 1,120.00
25 mg	￥ 1,960.00
50 mg	￥ 3,150.00
10mM * 1mL in DMSO	￥ 665.00

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生物活性

YM201636是PIKfyve的细胞渗透性和选择性抑制剂（IC50 = 33 nM）。

靶点信息

PIKfyve	p110α
33 nM	3.3 μM

溶解度 *

In vitro	DMSO	31 mg/mL (66.3 mM)
	Water	Insoluble
	Ethanol	Insoluble
* <1 mg/ml means slightly soluble or insoluble. * Please note that Adooq tests the solubility of all compounds in-house, and the actual solubility may differ slightly from published values. This is normal and is due to slight batch-to-batch variations.

制备储备液

Concentration / Solvent Volume / Mass	1 mg	5 mg	10 mg
0.1 mM	21.39 mL	106.95 mL	213.9 mL
0.5 mM	4.28 mL	21.39 mL	42.78 mL
1 mM	2.14 mL	10.7 mL	21.39 mL
5 mM	0.43 mL	2.14 mL	4.28 mL

*The above data is based on the productmolecular weight 467.5 . Batch specific molecular weights may vary from batch to batch due to solvent of hydration, which will affect the solvent volumes required to prepare stock solutions.

化学数据

目录号	A11064
作用机制	Inhibitor (抑制剂)
M. Wt	467.5
Formula	C25H21N7O3
Purity	>99%
Storage	Store lyophilized at -20ºC, keep desiccated. In lyophilized form, the chemical is stable for 36 months. In solution, store at -20ºC and use within 3 months to prevent loss of potency. Aliquot to avoid multiple freeze/thaw cycles.
CAS No.	371942-69-7
Synonyms	YM-201636
SMILES	C1COCCN1C2=NC(=NC3=C2OC4=C3C=CC=N4)C5=CC(=CC=C5)NC(=O)C6=CN=C(C=C6)N