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GPCR / G Protein

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Nebivolol

Catalog No. A13738
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Beta-1 adrenergic receptor blocker

Nebivolol是一种选择性抑制β-1肾上腺素能受体，IC50为0.8 nM。了解更多

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Doxazosin

Catalog No. A17779
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α-1 adrenergic receptor blocker

Doxazosin is an α-1 adrenergic receptor blocker that inhibits the binding of norepinephrine, which is released from sympathetic nerve terminals, to the α-1 receptors on the membrane of vascular smooth muscle cells. Blockages of the alpha-1 adrenergic action on the vascular smooth muscles lead to a decrease in vascular resistance and antihypertensive activity. 了解更多

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Metoprolol tartrate

Catalog No. A11713
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Beta1 receptor blocker

Metoprolol tartrate是一种选择性β1受体阻滞剂，用于治疗多种心血管系统疾病，尤其是高血压。了解更多

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Moxisylyte hydrochloride

Catalog No. A17725
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alpha-adrenergic blocking agent

Moxisylyte hydrochloride is an alpha-adrenergic blocking agent that is used in Raynaud's disease. It is also used locally in the eye to reverse the mydriasis caused by phenylephrine and other sympathomimetic agents. 了解更多

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Bisoprolol fumarate

Catalog No. A10149
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β1 adrenergic receptor blocker

Bisoprolol fumarate是一种属于β受体阻滞剂的药物，β受体阻滞剂是一类主要用于心血管疾病的药物。更具体地说，它是一种选择性的β1肾上腺素能受体阻滞剂。了解更多

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Phentolamine HCl

Catalog No. A13421
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α-Adrenergic blocker

Phentolamine HCl是一种AR(α肾上腺素能)阻滞剂。了解更多

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Pindolol

Catalog No. A13422
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Beta adrenergic receptor blocker

Pindolol是一种非选择性β阻断剂，具有部分β肾上腺素能受体激动剂活性。了解更多

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Esmolol

Catalog No. A17776
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β-adrenergic blocker

Esmolol is a short acting hyperselective β-adrenergic blocker effective in blunting adrenergic response to several perioperative stimuli and so it might interfere in the effect of the anesthetic drugs on the brain. 了解更多

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S(-)-Propranolol HCl

Catalog No. A13428
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β-adrenergic blocker

S(-)-Propranolol HCl是一种非选择性的β-肾上腺素能受体（βAR）拮抗剂，对β1AR和β2AR具有高亲和力，Ki值分别为1.8 nM和0.8 nM。盐酸普萘洛尔抑制[3H] -DHA与大鼠脑膜制剂的结合，IC50为12 nM。了解更多

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Orphenadrine citrate

Catalog No. A11712
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NMDA receptor 拮抗剂

Orphenadrine柠檬酸盐是NMDA受体拮抗剂，Ki为6.0μM，还是HERG钾离子通道阻断剂。了解更多

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Trimethobenzamide hydrochloride

Catalog No. A17648
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D2 receptor blocker

Trimethobenzamide hydrochloride is a blocker of the D2 receptor. Trimethobenzamide is an antiemetic used to prevent nausea and vomiting. 了解更多

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Dicarbine

Catalog No. A18925
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Dopamine receptor blocker

Dicarbine blocks dopamine receptors in various brain parts and prevents the depression of the conditioned defence reflexes caused by stimulation of the mesencephalic portion of the reticular formation. Dicarbine could be used to treat patients with schizophrenia and alcoholic psychosis in clinical. 了解更多

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