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GSK-269984A
Catalog No. A17096 -
CAY10471 Racemate
Catalog No. A11760 Prostaglandin D2 receptor CRTH2 antagonistCAY10471 Racemate (TM30089 Racemate) is a potent and highly selective prostaglandin D2 receptor CRTH2 antagonist. 了解更多 -
ONO-AE3-208
Catalog No. A11516 EP4 antagonistONO-AE3-208 is an EP4 antagonist, and suppresses cell invasion, migration, and metastasis of prostate cancer. 了解更多 -
MK-2894 sodium salt
Catalog No. A11498 EP4 antagonistMK-2894 sodium salt is a highly potent and selective second generation EP4 antagonist. 了解更多 -
Terutroban
Catalog No. A20884 thromboxane-prostaglandin receptor antagonistTerutroban is a thromboxane-prostaglandin receptor antagonist. 了解更多 -
CJ-42794
Catalog No. A21948 EP4 antagonistCJ-42794 is a selective prostaglandin E receptor subtype 4 (EP4) antagonist, inhibits [3H]-PGE2 binding to the human EP4 receptor with a mean pKi of 8.5, a binding affinity that was at least 200-fold more selective for the human EP4 receptor than other human EP receptor subtypes (EP1, EP2, and EP3). 了解更多 -
BAY-u 3405
Catalog No. A13751 -
MF498
Catalog No. A15532 -
PF-04418948
Catalog No. A12894 -
TG6-10-1
Catalog No. A15968 -
Grapiprant (CJ-023423)
Catalog No. A15964 prostaglandin EP4 receptor 拮抗剂Grapiprant (CJ-023423)是一种具有抗痛觉过敏特性的新型，有效且选择性的前列腺素EP4受体拮抗剂。 了解更多 -
A2A receptor antagonist 1
Catalog No. A12567 adenosine A2A/A1 receptor antagonistA2A receptor antagonist 1 (CPI-444 analog) is an antagonist of both adenosine A2A receptor and A1 receptor with Kis of 4 and 264 nM, respectively. 了解更多 -
Tonapofylline
Catalog No. A21328 adenosine A1 receptor antagonistTonapofylline (BG 9928) is an orally active and selective adenosine A1 receptor antagonist with a Ki of 7.4 nM for human adenosine A1 receptor (hA1), which displays 915-fold selectivity versus human adenosine A2A receptor and 12-fold selectivity versus human adenosine A2B receptor and is used in development for the treatment of heart failure. 了解更多 -
Rolofylline
Catalog No. A21649 adenosine A1 receptor antagonistRolofylline (KW-3902) is a potent, selective adenosine A1 receptor antagonist that is under development for the treatment of patients with acute congestive heart failure and renal impairment. 了解更多 -
Derenofylline
Catalog No. A21990 adenosine A1 receptor antagonistDerenofylline (SLV 320) is a potent, selective and orally active adenosine A1 receptor antagonist, with Ki values of 1 nM, 200 nM and 398 nM for human A1, A3 and A2A receptors respectively. 了解更多 -
Istradefylline (KW-6002)
Catalog No. A11451 -
SYN-115 (Tozadenant)
Catalog No. A11560 A2a receptor 拮抗剂SYN115是口服，有效和选择性的腺苷2a（A2a）受体抑制剂，作用于人类和恒河猴的 adenosine A2A 受体，Ki 值分别为 11.5 nM 和 6 nM。 了解更多 -
Aminophylline
Catalog No. A10066 Adenosine receptor 拮抗剂Aminophylline是一种非选择性的腺苷受体拮抗剂和磷酸二酯酶抑制剂，能够逆转局部缺血引起的bradyasystole。 了解更多 -
Dyphylline
Catalog No. A10339 Adenosine receptor 拮抗剂Dyphylline是黄嘌呤衍生物，具有支气管扩张药和血管扩张药的作用。 它充当腺苷受体拮抗剂和磷酸二酯酶抑制剂。 了解更多 -
SCH 442416
Catalog No. A12695 A2A Receptor 拮抗剂SCH 442416是一种选择性的腺苷A2A受体拮抗剂。以高亲和力结合人和大鼠A2A受体（Ki值分别为0.048和0.5 nM）。在体外对hA2A的选择性比hA1高> 23000倍，并且对hA2B和hA3受体的亲和力最小（IC50> 10μM）。 了解更多 -
CVT 6883
Catalog No. A13745 -
CF-102
Catalog No. A14402 -
CGS-15943
Catalog No. A14327 -
Preladenant
Catalog No. A13504 -
DPCPX
Catalog No. A16104 -
Vipadenant (BIIB-014)
Catalog No. A13963 A2A receptor 拮抗剂Vipadenant，也称为BIIB014，CEB-4520，是针对帕金森氏症的有效，选择性和口服腺苷A2A受体拮抗剂。Vipadenant在帕金森氏病的常用模型中显示出强大的口服活性。 了解更多 -
Theophylline-7-acetic acid
Catalog No. A16822 -
Proxyphylline
Catalog No. A16821 A1 adenosine receptors 拮抗剂Proxyphylline是茶碱的衍生物，由于其心血管特性而被用作支气管扩张剂。它与A2腺苷受体（对于血小板，Ki = 850μM）选择性拮抗A1腺苷受体（对于牛脑，Ki = 82 nM）。 了解更多 -
AZD-4635 (HTL1071)
Catalog No. A16820 -
MRS1177
Catalog No. A16871 -
MRS1186
Catalog No. A16870 -
CB1 antagonist 2
Catalog No. A18810 CB1 antagonistCB1 antagonist 2 is caimabinoid 1 (CB1) antagonist extracted from patent WO2016184310A1, compound 3, inhibits CB1 in vivo with an IC50 of 25.5 nM. 了解更多 -
(±)-Ibipinabant
Catalog No. A21439 CB-1 receptor antagonist(±)-Ibipinabant ((±)-SLV319) is the racemate of SLV319. (±)-Ibipinabant ((±)-SLV319) is a potent and selective cannabinoid-1 (CB-1) receptor antagonist with an IC50 of 22 nM. 了解更多 -
Taranabant racemate
Catalog No. A21699 CB1 antagonist/inverse agonistTaranabant racemate is an antagonist and/or inverse agonist of the Cannabinoid-1 (CB1) receptor extracted from patent WO 2004048317 A1. 了解更多 -
CP 945598 HCl (Otenabant HCl)
Catalog No. A11942 -
Otenabant
Catalog No. A15200
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