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GPCR / G Protein

产品 201 到 250 共 860个

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  1. Medetomidine HCl
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    Medetomidine HCl

    Catalog No. A13775
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    adrenergic alpha-2 receptor 激动剂
    Medetomidine Hydrochloride是一种肾上腺素α2-受体激动剂，Ki为1.08 nM，比作用于α1-adrenoceptor选择性高1620倍。由于其镇痛和镇静作用而被用于兽医学。 了解更多
  2. CL 316243 disodium salt
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    CL 316243 disodium salt

    Catalog No. A13657
    β3 adrenergic 激动剂
    CL 316243 disodium salt是一种3β-肾上腺素能激动剂，被开发为一种抗肥胖和糖尿病的药物，并使小鼠的血糖水平迅速下降。 了解更多
  3. BRL 37344 Na Salt
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    BRL 37344 Na Salt

    Catalog No. A13676
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    β3-adrenergic receptors 激动剂
    BRL 37344 Na Salt是具有脂解活性的β3-AR（β3-肾上腺素能受体）选择性激动剂。 了解更多
  4. Celiprolol HCl
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    Celiprolol HCl

    Catalog No. A13623
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    adrenergic receptor 拮抗剂
    Celiprolol HCl是一种b1肾上腺素能受体拮抗剂和b2肾上腺素能受体局部激动剂，在体外显示其ED50值为40-50 uM可使人的动脉和静脉松弛。 了解更多
  5. Guanabenz acetate
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    Guanabenz acetate

    Catalog No. A13635
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    2A-AR adrenergic 激动剂
    Guanabenz acetate是a2A-AR肾上腺素能激动剂和IGRS（咪唑啉I2结合位点）选择性配体。 了解更多
  6. BRL 44408 maleate
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    BRL 44408 maleate

    Catalog No. A13399
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    Adrenoceptors 拮抗剂
    BRL 44408 maleate是一种高纯度肾上腺素受体拮抗剂。它增加全身给药后海马去甲肾上腺素的释放。 了解更多
  7. Cimaterol
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    Cimaterol

    Catalog No. A13401
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    β-adrenergic receptors 激动剂
    Cimaterol是β的有效激动剂；肾上腺素能受体(人β的pEC50 = 8.13、8.78和6.62；1β，2β和3β)。 了解更多
  8. HEAT hydrochloride (BE 2254)
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    HEAT hydrochloride (BE 2254)

    Catalog No. A13408
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    Adrenergic α1 Receptor 拮抗剂
    HEAT hydrochloride (BE 2254)是一种选择性很强的α1-肾上腺素受体拮抗剂，是3-[125I]-衍生物的前体。肾上腺素受体或肾上腺素能受体是参与多种交感神经系统过程的G蛋白偶联受体。 了解更多
  9. Idazoxan Hydrochloride
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    Idazoxan Hydrochloride

    Catalog No. A13409
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    α2- adrenoceptor 拮抗剂 / I2 imidazoline receptor 激动剂
    Idazoxan hydrochloride 是α2-AR肾上腺素受体拮抗剂和潜在I2咪唑啉受体激动剂。还显示I1咪唑啉受体拮抗剂活性。(I1、I2和α的公钥基础设施值分别为5.90、7.22、8.01、7.43和7.7)。 了解更多
  10. JP 1302 2HCl
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    JP 1302 2HCl

    Catalog No. A13412
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    α2C 拮抗剂
    JP 1302 2HCl是一种强效和选择性α2C拮抗剂。 了解更多
  11. Phentolamine HCl
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    Phentolamine HCl

    Catalog No. A13421
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    α-Adrenergic blocker
    Phentolamine HCl是一种AR(α肾上腺素能)阻滞剂。 了解更多
  12. Rauwolscine
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    Rauwolscine

    Catalog No. A13426
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    α2-adrenergic receptor 拮抗剂
    Rauwolscine是一种天然生物碱，具有选择性和可逆性α2肾上腺素能受体拮抗剂(Ki = 12 nM)。 了解更多
  13. S-(-)-Atenolol
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    S-(-)-Atenolol

    Catalog No. A13427
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    Adrenoceptors 拮抗剂
    S-(-)-Atenolol是阿替洛尔的活性对映体，阿替洛尔是心脏选择性β肾上腺素能阻滞剂。 了解更多
  14. S(-)-Propranolol HCl
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    S(-)-Propranolol HCl

    Catalog No. A13428
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    β-adrenergic blocker
    S(-)-Propranolol HCl是一种非选择性的β-肾上腺素能受体（βAR）拮抗剂，对β1AR和β2AR具有高亲和力，Ki值分别为1.8 nM和0.8 nM。 盐酸普萘洛尔抑制[3H] -DHA与大鼠脑膜制剂的结合，IC50为12 nM。 了解更多
  15. (S)-Timolol maleate
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    (S)-Timolol maleate

    Catalog No. A13429
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    Adrenoceptors 拮抗剂
    (S)-Timolol maleate是对β有选择性肾上腺素能受体拮抗剂；β1-AR。 了解更多
  16. SR 59230A HCl
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    SR 59230A HCl

    Catalog No. A13430
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    Adrenoceptors 拮抗剂
    SR 59230A HCl是3β-肾上腺素受体拮抗剂。 了解更多
  17. Tulobuterol
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    Tulobuterol

    Catalog No. A13432
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    Adrenergic Receptor 激动剂
    Tulobuterol是β-肾上腺素能受体激动剂，在结构上与特布他林有关。 了解更多
  18. UK 14,304 tartrate
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    UK 14,304 tartrate

    Catalog No. A13433
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    Adrenoceptors 激动剂
    UK 14,304 tartrate是一种全α2肾上腺素能激动剂。 了解更多
  19. Xylazine HCl
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    Xylazine HCl

    Catalog No. A13434
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    Adrenergic Receptor 激动剂
    Xylazine hydrochloride是α2A-AR、α2B-AR和α2C-AR的活化剂。 了解更多
  20. Tamsulosin hydrochloride
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    Tamsulosin hydrochloride

    Catalog No. A14936
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    α1 receptor 拮抗剂
    Tamsulosin hydrochloride是一种选择性的α1受体拮抗剂，是用于良性前列腺增生的药物。 了解更多
  21. (R,R)-Formoterol
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    (R,R)-Formoterol

    Catalog No. A14964
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    β2-adrenoceptor 激动剂
    (R,R)-Formoterol是一种长效β2激动剂，用于哮喘和慢性阻塞性疾病的治疗。 了解更多
  22. Guanfacine hydrochloride
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    Guanfacine hydrochloride

    Catalog No. A15098
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    α2A-adrenoceptor 激动剂
    Guanfacine hydrochloride是一种抗高血压药，是一种选择性的α2A肾上腺素受体激动剂，Kd为31 nM，选择性是α2B肾上腺素受体的60倍。 了解更多
  23. HOKU-81
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    HOKU-81

    Catalog No. A15117
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    Metabolites of tulobuterol
    HOKU-81是新型支气管扩张剂，是妥洛特罗的代谢产物之一。 了解更多
  24. ICI-118551
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    ICI-118551

    Catalog No. A15878
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    β2 adrenergic receptor 拮抗剂
    ICI-118551是选择性的β2肾上腺素能受体（肾上腺素受体）拮抗剂。 了解更多
  25. Vilanterol trifenatate
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    Vilanterol trifenatate

    Catalog No. A15998
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    β2-adrenergic receptor 激动剂
    Vilanterol trifenatate是一种长效的β-2激动剂药物，于2013年5月与葛兰素氟替卡松合用，获葛兰素史克（Brax Elmitta）出售为Breo Ellipta，用于治疗慢性阻塞性肺疾病（COPD）。 了解更多
  26. TAK 259
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    TAK 259

    Catalog No. A16186
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    α1D Adrenoceptor 拮抗剂
    TAK-259是一种新型的，选择性的，口服活性的α1D肾上腺素受体拮抗剂（α1D，Ki = 1.1 nM），具有抗尿频效应并减少人类以太相关基因（hERG）的责任。 了解更多
  27. Brimonidine Tartrate
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    Brimonidine Tartrate

    Catalog No. A15033
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    α-adrenergic receptor 激动剂
    Brimonidine Tartrate是一种高度选择性的α-肾上腺素能受体激动剂，对α2A肾上腺素能受体的EC50为0.45 nM。 了解更多
  28. Acebutolol HCl
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    Acebutolol HCl

    Catalog No. A16387
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    β-adrenergic receptors 拮抗剂
    Acebutolol HCl是一种β-肾上腺素能受体拮抗剂，用于治疗高血压，心绞痛和心律不齐。 了解更多
  29. Clorprenaline HCl
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    Clorprenaline HCl

    Catalog No. A16465
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    β2-adrenergic receptor 激动剂
    Clorprenaline HCl是一种β2受体激动剂，具有显着的支气管扩张作用。 了解更多
  30. Vilanterol
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    Vilanterol

    Catalog No. A13125
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    ultra-long-acting β? adrenoreceptor 激动剂
    Vilanterol是一种新的选择性β2-AR激动剂，PEC50值为10.37±0.05。 了解更多
  31. Urapidil
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    Urapidil

    Catalog No. A17074
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    α1 adrenoreceptor 拮抗剂
    Urapidil是一种α1肾上腺素受体拮抗剂和5-HT1A受体激动剂。 了解更多
  32. Methoxamine HCl
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    Methoxamine HCl

    Catalog No. A17365
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    alpha-1 adrenergic agonist
    Methoxamine Hydrochloride is an alpha-1 adrenergic agonist that causes prolonged peripheral vasoconstriction. 了解更多
  33. Nifenalol HCl
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    Nifenalol HCl

    Catalog No. A17246
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    beta-adrenergic receptor antagonist
    Nifenalol, also known as INPEA, is a new beta-adrenergic receptor antagonist. 了解更多
  34. Ractopamine HCl
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    Ractopamine HCl

    Catalog No. A17372
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    beta-Adrenergic agonist
    Ractopamine HCl is a beta-Adrenergic agonist. It acts by being a full agonist at the TAAR1. 了解更多
  35. Moxisylyte hydrochloride
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    Moxisylyte hydrochloride

    Catalog No. A17725
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    alpha-adrenergic blocking agent
    Moxisylyte hydrochloride is an alpha-adrenergic blocking agent that is used in Raynaud's disease. It is also used locally in the eye to reverse the mydriasis caused by phenylephrine and other sympathomimetic agents. 了解更多
  36. Midodrine hydrochloride
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    Midodrine hydrochloride

    Catalog No. A17757
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    Adrenergic alpha-1 agonist
    Midodrine hydrochloride is an ethanolamine derivative that is an adrenergic alpha-1 agonist. It is used as a vasoconstrictor agent in the treatment of hypotension. It improves clinical outcome of chronic hypotension. 了解更多
  37. Midodrine
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    Midodrine

    Catalog No. A17758
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    adrenergic alpha-1 agonist
    Midodrine is an ethanolamine derivative that is an adrenergic alpha-1 agonist. It is used as a vasoconstrictor agent in the treatment of HYPOTENSION. 了解更多
  38. Fenoterol
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    Fenoterol

    Catalog No. A17774
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    Beta 2 adrenergic agonist
    Fenoterol is a Beta 2 adrenergic agonist designed to open up the airways to the lungs. It is classed as sympathomimetic beta agonist and asthma medication. 了解更多
  39. Esmolol
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    Esmolol

    Catalog No. A17776
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    β-adrenergic blocker
    Esmolol is a short acting hyperselective β-adrenergic blocker effective in blunting adrenergic response to several perioperative stimuli and so it might interfere in the effect of the anesthetic drugs on the brain. 了解更多
  40. Doxazosin
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    Doxazosin

    Catalog No. A17779
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    α-1 adrenergic receptor blocker
    Doxazosin is an α-1 adrenergic receptor blocker that inhibits the binding of norepinephrine, which is released from sympathetic nerve terminals, to the α-1 receptors on the membrane of vascular smooth muscle cells. Blockages of the alpha-1 adrenergic action on the vascular smooth muscles lead to a decrease in vascular resistance and antihypertensive activity. 了解更多
  41. Brimonidine
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    Brimonidine

    Catalog No. A17899
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    α2-adrenergic receptor agonist
    Brimonidine (UK 14304) is a full α2-adrenergic receptor (α2-AR) agonist. 了解更多
  42. Nylidrin Hydrochloride
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    Nylidrin Hydrochloride

    Catalog No. A17947
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    beta-adrenergic agonist
    Nylidrin hydrochloride is a beta-adrenergic agonist. Nylidrin hydrochloride is shown to be an effective inhibitor of IgE-mediated release of histamine from human basophils, and thus can be used as antiallergic agent. 了解更多
  43. Metipranolol hydrochloride
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    Metipranolol hydrochloride

    Catalog No. A18064
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    β-adrenergic receptor antagonist
    Metipranolol (hydrochloride) is a non-selective β-adrenergic receptor (β-AR) antagonist. Formulations containing metipranolol have been used in the treatment of elevated IOP in patients with ocular hypertension or glaucoma. 了解更多
  44. Anisodamine
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    Anisodamine

    Catalog No. A18215
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    alpha-1 adrenergic receptors / mAChRs inhibitor
    Anisodamine is an inhibitor of alpha-1 adrenergic receptors and mAChRs isolated from Chinese solanacea plant. 了解更多
  45. Tulobuterol hydrochloride
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    Tulobuterol hydrochloride

    Catalog No. A18226
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    β2-adrenergic receptor agonist
    Tulobuterol Hydrochloride is a long-acting beta2-adrenergic receptor agonist. 了解更多
  46. BI-167107
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    BI-167107

    Catalog No. A18687
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    β2 adrenergic receptor agonist
    BI-167107 is a high affinity, full agonist that binds to the β2 adrenergic receptor (β2AR) with a dissociation constant Kd of 84 pM. 了解更多
  47. Atenolol
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    Atenolol

    Catalog No. A21962
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    β1 receptor antagonist
    Atenolol is a selective β1 receptor antagonist. 了解更多
  48. H4 Receptor antagonist 1
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    H4 Receptor antagonist 1

    Catalog No. A18929
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    histamine H4 receptor inverse agonist
    H4 Receptor antagonist 1 is a potent and selective histamine H4 receptor inverse agonist, with an IC50 of 19 nM. 了解更多
  49. Chlorcyclizine hydrochloride
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    Chlorcyclizine hydrochloride

    Catalog No. A18025
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    histamine H1 antagonist
    Chlorcyclizine hydrochloride is a histamine H1 antagonist. 了解更多
  50. Toreforant
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    Toreforant

    Catalog No. A21058
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    histamine H4 receptor (H4R) antagonist
    Toreforant is a potent and selective histamine H4 receptor (H4R) antagonist, with a Ki at the human receptor of 8.4 nM. 了解更多

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  1. 5-HT Receptors (143)
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  10. G Protein (26)
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  1. Inhibitor (抑制剂) (86)
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  13. Histamine H1 receptor (1)
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