GPCR / G Protein
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LY 344864 S-enantiomer
Catalog No. A21742 5-HT1F receptor agonistLY 344864 S-enantiomer is the S-enantiomer of LY344864. LY344864 is a 5-HT1F receptor agonist. 了解更多 -
LY 344864 hydrochloride
Catalog No. A21748 5-HT1F agonistLY 344864 hydrochloride is a selective 5-HT1F agonist with a Ki of 6 nM. 了解更多 -
Vilazodone D8
Catalog No. A21876 SSR inhibitor / 5-HT1A receptor partial agonistVilazodone D8 is the a deuterium labeled vilazodone, which is a combined serotonin specific reuptake inhibitor (SSRI) and 5-HT1A receptor partial agonist. 了解更多 -
SB-269970 hydrochloride
Catalog No. A21889 5-HT7 receptor antagonistSB269970 hydrochloride (SB-269970A) is a hydrochloride salt form of SB-269970, which is a 5-HT7 receptor antagonist with the pKi of 8.3, exhibits >50-fold selectivity against other receptors. 了解更多 -
SB-224289 hydrochloride
Catalog No. A21920 5-HT1B receptor antagonistSB-224289 hydrochloride is a selective 5-HT1B receptor antagonist, with anxiolytic effect. 了解更多 -
Ritanserin
Catalog No. A21976 5-HT2 receptor antagonistRitanserin (R 55667) is a highly potent, relatively selective, orally active, long acting antagonist of 5-HT2 receptor, with an IC50 of 0.9 nM, less active on Histamine H1, Dopamine D2, Adrenergic α1, Adrenergic α2 receptors. 了解更多 -
Eplivanserin mixture
Catalog No. A21987 serotonin reuptake inhibitor/5-HT2A receptor antagonistEplivanserin mixture is a selective serotonin reuptake inhibitor and a 5-HT2A receptor antagonist, extracted from patent WO 2005/002578 A1. 了解更多 -
Ziprasidone D8
Catalog No. A21989 5-HT / dopamine receptor antagonistZiprasidone D8 is deuterium labeled Ziprasidone, which is a combined 5-HT (serotonin) and dopamine receptor antagonist which exhibits potent effects of antipsychotic activity. 了解更多 -
Aripiprazole (D8)
Catalog No. A22004 human 5-HT1A receptor partial agonistAripiprazole D8 (OPC-14597 D8) is the deuterium labeled Aripiprazole, which is a human 5-HT1A receptor partial agonist with a Ki of 4.2 nM. 了解更多