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GPCR / G Protein

产品 301 到 350 共 860个

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  1. Etizolam
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    Etizolam

    Catalog No. A14257
    PAFR 拮抗剂
    Etizolam是一种具有抗焦虑活性的特异性血小板活化因子（PAF）拮抗剂。 了解更多
  2. YM-264
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    YM-264

    Catalog No. A20139
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    PAF 拮抗剂
    YM-264 is a selective, potent and orally active platelet-activating factor (PAF) antagonist with a pKi value of 8.85 for rabbit platelet membranes. 了解更多
  3. 48740 RP
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    48740 RP

    Catalog No. A12339
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    PAF 拮抗剂
    48740 RP (RP-55778) is a platelet-activating factor (PAF) antagonist. 了解更多
  4. Aglafoline
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    Aglafoline

    Catalog No. A12257
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    PAF antagonist
    Aglafoline is an effective PAF antagonist not only in vitro, but also in vivo. 了解更多
  5. Foropafant
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    Foropafant

    Catalog No. A13388
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    PAF receptor antagonist
    Foropafant (SR27417) highly potent, competitive, selective and orally active antagonist of platelet-activating factor (PAF) receptor. 了解更多
  6. CP-96486
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    CP-96486

    Catalog No. A12471
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    LTD4/PAF receptor antagonist
    CP-96486 is a potent and orally active leukotriene D4 (LTD4)/platelet activating factor (PAF) receptor antagonist with Kis of 20 and 24 nM, respectively. 了解更多
  7. QS 11
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    QS 11

    Catalog No. A11228
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    ATPase and GTPase 抑制剂
    QS-11是ADP-核糖基化因子1（ARFGAP1）抑制剂的GTPase活化蛋白。 了解更多
  8. CCG-63802
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    CCG-63802

    Catalog No. A11373
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    CCG-63802是G蛋白信号(RGS)蛋白调节因子的可逆抑制剂。在RGS蛋白中具有选择性，在RGS4中具有最大效力。 了解更多
  9. CASIN
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    CASIN

    Catalog No. A12912
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    Cdc42 GTPase 抑制剂
    CASIN是一种新型有效的Cdc42抑制剂。 了解更多
  10. CCG 50014
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    CCG 50014

    Catalog No. A16432
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    RGS4 抑制剂
    CCG 50014是RGS4的有效和选择性抑制剂，IC50为30 nM。 了解更多
  11. MK-6892
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    MK-6892

    Catalog No. A12982
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    GPR109A 激动剂
    MK-6892是高亲和力烟酸（NA）受体GPR109A的有效，选择性和完全激动剂。人GPR109A的MK-6892的Ki和GTPγSEC 50分别为4 nM和16 nM。 了解更多
  12. CID16020046
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    CID16020046

    Catalog No. A16818
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    GPR55 拮抗剂
    CID16020046是一种选择性的GPR55拮抗剂，在酵母中抑制GPR55的组成活性，IC50为150 nM。它对其他广谱GPCRs、离子通道、激酶和核受体表现出弱活性。 了解更多
  13. TM N1324
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    TM N1324

    Catalog No. A17038
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    GPR39 激动剂
    TM N1324是G蛋白偶联受体39（GPR39）的激动剂，在Zn2+存在下的EC50为9 nM/5 nM，而对于人/鼠GPR39，则在Zn2+不存在时的EC50为280 nM/180 nM。 了解更多
  14. GW-1100
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    GW-1100

    Catalog No. A11445
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    GPR40 antagonist
    GW-1100 is a selective GPR40 antagonist with a pIC50 of 6.9. 了解更多
  15. DJ-V-159
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    DJ-V-159

    Catalog No. A18853
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    GPRC6A agonist
    DJ-V-159 is an agonist for G protein-coupled receptor family C group 6 member A (GPRC6A). 了解更多
  16. GPR4 antagonist 1
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    GPR4 antagonist 1

    Catalog No. A12340
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    GPR4 antagonist
    GPR4 antagonist 1 is a GPR4 antagonist, with an IC50 of 189 nM. 了解更多
  17. G15
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    G15

    Catalog No. A13675
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    GPER/GPR30 antagonist
    G15 is a high affinity and selective G-protein-coupled estrogen receptor (GPER/GPR30) antagonist with a Ki of 20 nM. 了解更多
  18. LY2922470
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    LY2922470

    Catalog No. A12181
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    GPR40 agonist
    LY2922470 is a potent, selective and orally available agonist of the G protein-coupled receptor 40 (GPR40), with EC50s of 7 nM, 1 nM and 3 nM for human GPR40, mouse GPR40 and rat GPR40, respectively. 了解更多
  19. PSN632408
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    PSN632408

    Catalog No. A20902
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    GPR119 receptors agonist
    PSN632408 is an optimized agonist of GPR119 receptors that shows similar potency to OEA at both recombinant mouse and human GPR119 receptors, exhibiting EC50 values of 5.6 and 7.9 uM, respectively. 了解更多
  20. GPR40 Activator 1
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    GPR40 Activator 1

    Catalog No. A21154
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    GPR40 activator
    GPR40 Activator 1 is a potent GPR40 activator for treatment of type 2 diabetes. 了解更多
  21. GLPG0974
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    GLPG0974

    Catalog No. A21466
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    FFA2/GPR43 antagonist
    GLPG0974 is a free fatty acid receptor-2 (FFA2/GPR43) antagonist with an IC50 of 9 nM. 了解更多
  22. AM-1638
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    AM-1638

    Catalog No. A21505
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    GPR40/FFA1 full agonist
    AM-1638 is a potent and orally bioavailable GPR40/FFA1 full agonist with an EC50 of 0.16 μM. 了解更多
  23. AF64394
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    AF64394

    Catalog No. A21574
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    GPR3 inverse agonist
    AF64394 is a GPR3 inverse agonist, with a pIC50 of 7.3. 了解更多
  24. GPR40 Activator 2
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    GPR40 Activator 2

    Catalog No. A21642
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    GPR40 activator
    GPR40 Activator 2 is a potent GPR40 activator from patents WO 2012147516 A1, WO 2012046869A1 and WO 2011078371 A1. 了解更多
  25. (1R,2R)-2-PCCA(hydrochloride)
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    (1R,2R)-2-PCCA(hydrochloride)

    Catalog No. A21655
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    GPR88 receptor agonist
    (1R,2R)-2-PCCA hydrochloride is a diastereomer of 2-PCCA, and acts as a potent GPR88 receptor agonist, with an EC50 of 3 nM in cell-free assay, and 603 nM in cell assay. 了解更多
  26. AM-4668
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    AM-4668

    Catalog No. A21778
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    GPR40 agonist
    AM-4668 is a GPR40 agonist for type 2 diabetes. EC50s of 3.6 nM and 36 nM for GPR40 in A9 cells (GPR40 IP3 assay) and CHO cells (GPR40 aequorin assay), respectively. 了解更多
  27. AMG 837 sodium salt
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    AMG 837 sodium salt

    Catalog No. A21793
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    GPR40 agonist
    AMG 837 sodium salt is a potent GPR40 agonist(EC50=13 nM) with a superior pharmacokinetic profile and robust glucose-dependent stimulation of insulin secretion in rodents. 了解更多
  28. MK-0354
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    MK-0354

    Catalog No. A22008
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    GPR109a receptor agonist
    MK-0354 is a partial agonist of GPR109a receptor, for hGPR109a/ mGPR109a with EC50 of 1.65/1.08 μM, showed no activation of GPR109b. 了解更多
  29. AMG 837
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    AMG 837

    Catalog No. A21160
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    GPR40 agonist
    AMG 837 is a potent GPR40 agonist(EC50=13 nM) with a superior pharmacokinetic profile and robust glucose-dependent stimulation of insulin secretion in rodents. 了解更多
  30. Plerixafor 8HCl (DB06809)
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    Plerixafor 8HCl (DB06809)

    Catalog No. A10913
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    CXCR4 拮抗剂
    Plerixafor 8HCl (DB06809)是CXCR4趋化因子受体拮抗剂，作用于CXCR4和CXCL12介导调节的趋化性， IC50分别为44 nM和5.7 nM。 了解更多
  31. AMD 070
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    AMD 070

    Catalog No. A11315
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    CXCR4 拮抗剂
    AMD 070是CXCR4趋化因子受体拮抗剂。 了解更多
  32. AMD 3465 Hexahydrobromide
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    AMD 3465 Hexahydrobromide

    Catalog No. A11953
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    CXCR4 拮抗剂
    AMD 3465 Hexahydrobromide是一种有效的选择性CXCR4拮抗剂。 了解更多
  33. SRT3109
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    SRT3109

    Catalog No. A11097
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    CXCR2 ligand
    SRT3109是一种CXCR2配体，用于治疗趋化因子介导的疾病和状况。 了解更多
  34. WZ811
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    WZ811

    Catalog No. A12588
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    CXCR4 拮抗剂
    WZ811是4型C-X-C趋化因子受体（CXCR4）拮抗剂（EC50 = 0.3 nM）。在体外抑制CXCR4/基质细胞衍生因子1（SDF-1）介导的cAMP调节（EC50 = 1.2 nM）。 了解更多
  35. MSX-122
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    MSX-122

    Catalog No. A12596
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    CXCR4 抑制剂
    MSX-122是口服可生物利用的CXCR4抑制剂（IC50 =?10 nM），具有潜在的抗肿瘤和抗病毒活性。CXCR4抑制剂MSX-122与趋化因子受体CXCR4结合，阻止基质衍生因子-1（SDF-1）与CXCR4受体和受体激活结合，这可能导致肿瘤细胞增殖和迁移减少。 了解更多
  36. SRT3190
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    SRT3190

    Catalog No. A11577
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    SIRT1 activator
    SRT3190是一种强效cxcr2配体。 了解更多
  37. Reparixin
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    Reparixin

    Catalog No. A12383
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    CXCL8/CXCR1/2 抑制剂
    Reparixin是两种CXCL8受体CXCR1/2的有效抑制剂，它抑制CXCR2介导的细胞迁移（IC50 = 100 nM），而它强烈地阻断CXCR1介导的趋化性（IC50 = 1 nM）。 了解更多
  38. AMD3100 (Plerixafor)
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    AMD3100 (Plerixafor)

    Catalog No. A13074
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    CXCR4 拮抗剂
    AMD3100 (Plerixafor)是用于增殖造血干细胞的免疫刺激剂，并且是用于动员造血干细胞进行移植的趋化因子受体-4拮抗剂。 了解更多
  39. SCH-527123 (Navarixin)
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    SCH-527123 (Navarixin)

    Catalog No. A11555
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    CXCR1/CXCR2 拮抗剂
    SCH-527123 (Navarixin)是人CXCR1和CXCR2受体的强效选择性拮抗剂，IC50分别为42 nM和3 nM。 了解更多
  40. SB265610
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    SB265610

    Catalog No. A14195
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    CXCR2 拮抗剂
    SB265610是CXCR2 (Kd = 2.51 nM)的非肽变构反向激动剂，通过与不同于激动剂结合位点的区域结合来防止受体活化。它不与相关CXCR1受体结合。在体外和高氧诱导肺损伤的大鼠模型中，它已被证明能防止中性粒细胞趋化性。 了解更多
  41. SB225002
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    SB225002

    Catalog No. A14209
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    CXCR2 拮抗剂
    SB225002是一种有效的选择性CXCR2拮抗剂，IC50为22 nM，可抑制白介素IL-8与CXCR2的结合，选择性是其他测试的7-TMR的150倍以上。 了解更多
  42. Reparixin L-lysine salt
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    Reparixin L-lysine salt

    Catalog No. A15219
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    CXCL8 receptor 抑制剂
    Reparixin L-lysine salt是CXCL8受体的抑制剂，也抑制CXCR1和CXCR2的活化，已显示在各种损伤模型中减弱了炎症反应。 了解更多
  43. AMD-070 HCl
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    AMD-070 HCl

    Catalog No. A14997
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    CXCR4 拮抗剂
    在CXCR4 125I-SDF抑制结合试验中，AMD-070 HCl是一种有效的选择性CXCR4拮抗剂，IC50值为13 nM，抑制T-4型HIV-1（NL4.3株）在MT-4细胞中的复制和PBMC。 了解更多
  44. UNBS5162
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    UNBS5162

    Catalog No. A15439
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    CXCL chemokines 拮抗剂
    UNBS5162是一种新型萘二甲酰亚胺，可降低实验性前列腺癌中CXCL趋化因子的表达。9种癌细胞系的平均抗增殖活性IC50值为17.9 uM；UNBS3157的水解产物。 了解更多
  45. ATI-2341
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    ATI-2341

    Catalog No. A16351
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    CXCR4 激动剂
    ATI-2341是针对C-X-C趋化因子受体4型（CXCR4）（EC50 = 194 nM）的pepducin，是一种变构激动剂，可激活抑制性异三聚体G蛋白（Gi），从而促进cAMP生成的抑制并诱导钙动员。 了解更多
  46. NSC-23026
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    NSC-23026

    Catalog No. A17151
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    CXCR4 receptor modulator
    NSC-23026是CXCR4受体调节剂。 了解更多
  47. MSX-130
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    MSX-130

    Catalog No. A17150
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    CXCR4 拮抗剂
    MSX-130是CXCR4拮抗剂。 了解更多
  48. USL311
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    USL311

    Catalog No. A18778
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    CXCR4 拮抗剂
    USL311 is a CXCR4 receptor antagonist which prevents the binding of stromal-cell derived factor-1 (SDF-1 or CXCL12) to CXCR4. 了解更多
  49. Kynurenic acid
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    Kynurenic acid

    Catalog No. A16581
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    GPR35/CXCR8 拮抗剂
    Kynurenic acid, an endogenous tryptophan metabolite, is a broad-spectrum antagonist targeting NMDA, glutamate, α7 nicotinic acetylcholine receptor. Kynurenic acid is also an agonist of GPR35/CXCR8. 了解更多
  50. PS372424
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    PS372424

    Catalog No. A19421
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    Human CXCR3 拮抗剂
    PS372424, a three amino-acid fragment of CXCL10, is a specific human CXCR3 agonist with anti-inflammatory activity, which inhibits the binding of CXCR3 ligand CXCL10 to CXCR3 receptor with IC50 of 42 nM. 了解更多

产品 301 到 350 共 860个

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  1. 5-HT Receptors (143)
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