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LY 344864
Catalog No. A15148 -
Pimavanserin (ACP-103)
Catalog No. A14434 5-HT2A receptor 激动剂Pimavanserin (ACP-103)是一种有效的选择性5-HT2A受体反向激动剂，在基于细胞的功能测定中，平均pIC50为8.7。 了解更多 -
WAY 181187
Catalog No. A14163 -
Donitriptan
Catalog No. A13145 5-HT1B/1D receptors agonistDonitriptan is a potent, high efficacy agonist at 5-HT1B/1D receptors with pKis of 9.4 and 9.3, respectively. 了解更多 -
PRX933 hydrochloride
Catalog No. A12261 5-HT2c receptor agonistPRX933 hydrochloride is a 5-HT2c receptor agonist extracted from patent WO 2014140631 A1. 了解更多 -
Lesopitron dihydrochloride
Catalog No. A12950 5-HT1A receptor agonistLesopitron dihydrochloride is a full and selective 5-HT1A receptor agonist with IC50 of 125 nM in rat hippocampal membranes. 了解更多 -
WAY 163909
Catalog No. A21282 5-HT(2C) receptor agonistWAY 163909 is a potent and selective 5-HT(2C) receptor agonist with a Ki of 10.5??1.1 nM. 了解更多 -
Nelotanserin
Catalog No. A21506 5-HT2A inverse agonistNelotanserin is a potent 5-HT2A inverse agonist, a moderately potent 5-HT2C partial inverse agonist and a weak 5-HT2B inverse agonist, with IC50s of 1.7, 79, 791 nM in IP accumulation assays, respectively. 了解更多 -
LY 344864 S-enantiomer
Catalog No. A21742 5-HT1F receptor agonistLY 344864 S-enantiomer is the S-enantiomer of LY344864. LY344864 is a 5-HT1F receptor agonist. 了解更多 -
LY 344864 hydrochloride
Catalog No. A21748 5-HT1F agonistLY 344864 hydrochloride is a selective 5-HT1F agonist with a Ki of 6 nM. 了解更多 -
Vilazodone D8
Catalog No. A21876 SSR inhibitor / 5-HT1A receptor partial agonistVilazodone D8 is the a deuterium labeled vilazodone, which is a combined serotonin specific reuptake inhibitor (SSRI) and 5-HT1A receptor partial agonist. 了解更多 -
Aripiprazole (D8)
Catalog No. A22004 human 5-HT1A receptor partial agonistAripiprazole D8 (OPC-14597 D8) is the deuterium labeled Aripiprazole, which is a human 5-HT1A receptor partial agonist with a Ki of 4.2 nM. 了解更多 -
Mosapride citrate
Catalog No. A10607 -
Tianeptine sodium
Catalog No. A10931 -
BMY 7378
Catalog No. A11208 -
Prucalopride
Catalog No. A11771 5-HT Receptor 激动剂Prucalopride是一种选择性的，高亲和力的5-HT4受体激动剂，作用于5-HT4A和5-HT4B受体，Ki分别为2.5 nM和8 nM，比作用于5-HT受体亚型选择性高290倍以上。 了解更多 -
Clomipramine HCl
Catalog No. A10231 5-HT Receptor 激动剂Clomipramine HCl是下列转运蛋白的阻滞剂：5-羟色胺转运蛋白 (SERT)(Ki = 0.14 nM)，去甲肾上腺素转运蛋白（NET）(Ki = 54 nM)，多巴胺转运蛋白（DAT）(Ki = 3，020 nM)，甘氨酸转运蛋白（GlyT/LeuT）。 了解更多 -
Almotriptan malate (Axert)
Catalog No. A11799 5-HT Receptor 激动剂Almotriptan malate (Axert)是一种选择性的5-羟色胺1B/1D（5-HT1B/1D）受体激动剂，用于治疗成人偏头痛。 了解更多 -
Aripiprazole (Abilify)
Catalog No. A11801 5-HT1A receptor 激动剂Aripiprazole (Abilify)是人5-HT1A受体部分激动剂，Ki为4.2 nM。 了解更多 -
Eletriptan hydrobromide
Catalog No. A11418 5-HT1B/1D receptor 激动剂Eletriptan hydrobromide是一种选择性SR-1B/SR-1D激动剂。 了解更多 -
Lorcaserin
Catalog No. A12378 -
lorcaserin hydrochloride (APD-356)
Catalog No. A12598 serotonin 2C receptor 激动剂lorcaserin hydrochloride (APD-356)是血清素2C受体激动剂，可指示与减少热量饮食和增加体育锻炼以减轻慢性体重成人管理。 了解更多 -
RU 24969 hemisuccinate
Catalog No. A13833 5-HT1A/1B and 5-HT2C 激动剂RU 24969 hemisuccinate是有效的5-HT1A/1B和中度5-HT2C激动剂，也可能释放5-HT。 了解更多 -
S 32212 HCl
Catalog No. A13501 -
Eptapirone
Catalog No. A15923 5HT(1A) receptor 激动剂Eptapirone是一种有效的，选择性的，高效的5-HT1A受体激动剂，具有显着的抗焦虑和抗抑郁潜力。 了解更多 -
Pimavanserin
Catalog No. A15884 Serotonin2A Receptor Inverse 激动剂Pimavanserin是一种有效的选择性5-羟色胺5-HT2A反向激动剂，pIC50为8.73，用于治疗与帕金森氏病有关的精神病。 了解更多 -
Buspirone HCl
Catalog No. A15687 5HT(1A) receptor 激动剂Buspirone hydrochloride是一种具有5-D（2）多巴胺能作用的血清素能（5HT（1A）受体激动剂）抗焦虑药，用于焦虑症。 了解更多 -
Temanogrel
Catalog No. A17094 5-HT(2A) receptor 激动剂Temanogrel，也称为APD791，是一种高度选择性的5-羟基色胺2A受体反向激动剂，正在开发中，用于治疗动脉血栓形成。 了解更多 -
LY 344864 racemate
Catalog No. A17015 -
Eptapirone (F-11440)
Catalog No. A18338 5-HT1A receptor agonistEptapirone is a potent, selective, high efficacy 5-HT1A receptor agonist with marked anxiolytic and antidepressant potential. The affinity of F 11440 for 5-HT1A binding sites (pKi, 8.33) was higher than that of buspirone (pKi, 7.50), and somewhat lower than that of flesinoxan (pKi, 8.91). In vivo, F 11440 was 4- to 20-fold more potent than flesinoxan, and 30- to 60-fold more potent than buspirone. 了解更多 -
Norepinephrine
Catalog No. A11306 β1-selective adrenergic receptor agonistNorepinephrine (Levarterenol; L-Noradrenaline) is a β1-selective adrenergic receptor agonist with EC50 of 5.37 μM. 了解更多 -
AGN 192836
Catalog No. A13013 α2 adrenergic agonistAGN 192836 is a potent and selective α2 adrenergic agonist with EC50s of 8.7, 41 and 6.6 nM for α2A, α2B and α2C receptor, respectively. 了解更多 -
β3-AR agonist 1
Catalog No. A12777 β3-adrenergic receptor agonistβ3-AR agonist 1 (compound 15) is a highly potent, selective, and orally available β3-adrenergic receptor (β3-AR) agonist (EC50=18 nM), being inactive to β1-, β2-, and α1A-AR (β1/β3, β2/β3, and α1A/β3>556-fold). 了解更多 -
Norepinephrine hydrochloride
Catalog No. A21605 β1-selective adrenergic receptor agonistNorepinephrine hydrochloride (Levarterenol hydrochloride; L-Noradrenaline hydrochloride) is a β1-selective adrenergic receptor agonist with EC50 of 5.37 μM. 了解更多 -
Synephrine (Oxedrine)
Catalog No. A10882 -
Salbutamol sulfate (Albuterol)
Catalog No. A10819 Adrenergic Receptor 激动剂Salbutamol sulfate (Albuterol)是一种短效β2肾上腺素能受体激动剂。 了解更多 -
Phenylephrine HCl
Catalog No. A11666 α1-adrenergic receptor 激动剂Phenylephrine HCl是一种选择性的α1肾上腺素能受体激动剂，主要用作减充血剂，扩张瞳孔和增加血压的药物。 了解更多 -
Isoprenaline HCl
Catalog No. A10484 β adrenoceptor 激动剂Isoprenaline HCl或isoproterenol是非选择性β肾上腺素能激动剂，在结构上类似于肾上腺素。 了解更多 -
Detomidine hydrochloride
Catalog No. A10298 Adrenergic Receptor 激动剂Detomidine hydrochloride是具有镇痛作用的镇静剂。α2-肾上腺素能激动剂产生剂量依赖性的镇静和镇痛作用，并通过激活α2儿茶酚胺受体介导，从而引起负反馈反应，从而减少兴奋性神经递质的产生。 了解更多 -
Clonidine hydrochloride
Catalog No. A10232 Alpha adrenergic 激动剂Clonidine hydrochloride被归类为中枢作用的α肾上腺素能激动剂。Clonidine主要作为咪唑啉受体激动剂。 了解更多 -
Dobutamine hydrochloride
Catalog No. A10325 Adrenoceptors 激动剂Dobutamine hydrochloride是一种直接作用剂，其主要活性来自刺激心脏的β1肾上腺素能受体，增加收缩力和心输出量。 了解更多
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