A-9758
目录号: A19078
RORγt inverse 激动剂
A-9758 是一种 RORγ 配体,同时是一种高效、选择性的 RORγt 反向激动剂(IC50=5 nM),并且对 IL-17A 的释放显示出强大的效力。
Discription | A-9758 is a RORγ ligand and a potent, selective RORγt inverse agonist (IC50=5 nM), and exhibits robust potency against IL-17A release. | ||
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目录号 | A19078 |
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分子式 | C25H23Cl2F3N2O3 |
分子量 | 527.36 |
CAS号 | 2055271-22-0 |
SMILES | O=C(C1CCN(C(C2=CC=C(Cl)C(CC(N3C)=CC4=C3C=C(C(F)(F)F)C=C4C)=C2Cl)=O)CC1)O |
其他名称 | A9758, A 9758 |
储存条件 | Store lyophilized at -20ºC, keep desiccated. |
Calculate the dilution required to prepare a stock solution. This equation is commonly abbreviated as: C1V1 = C2V2