AGN 205728
目录号: A16296
RARγ 拮抗剂
AGN 205728 是一种强效且选择性的 RARγ 拮抗剂,其 Ki/IC95 值为 3 nM/0.6 nM;对 RARα 和 RARβ 无抑制作用。
Discription | AGN 205728 is a potent and selective RARγ antagonist with Ki/IC95 values of 3 nM/ 0.6 nM; no inhibiton on RARα and RARβ. |
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目录号 | A16296 |
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分子式 | C29H27NO3 |
分子量 | 437.53 |
CAS号 | 859498-05-8 |
SMILES | CC1=CC=C(C=C1)C2=CCC(C)(C)C3=C2C=CC(=C3)/C(=N/O)/C=C/C4=CC=C(C=C4)C(=O)O |
其他名称 | AGN205728, AGN-205728 |
储存条件 | Store lyophilized at -20ºC, keep desiccated. |
Calculate the dilution required to prepare a stock solution. This equation is commonly abbreviated as: C1V1 = C2V2