Almorexant
目录号: A12503
OX Ant激动剂
Almorexant(ACT078573)是一种强效且具有竞争性的双重俄罗斯素1受体(OX1)/俄罗斯素2受体(OX2)拮抗剂,其Ki值分别为OX1的1.3 nM和OX2的0.17 nM。
Discription | Almorexant(ACT078573) is a potent and competitive dual orexin 1 receptor (OX1)/orexin 2 receptor (OX2) antagonist with Ki values of 1.3 and 0.17 nM for OX1 and OX2, respectively. | |||||
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Targets |
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Cell Research |
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目录号 | A12503 |
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分子式 | C29H31F3N2O3 |
分子量 | 512.56 |
CAS号 | 871224-64-5 |
SMILES | CNC(=O)[C@@H](C1=CC=CC=C1)N2CCC3=CC(=C(C=C3[C@@H]2CCC4=CC=C(C=C4)C(F)(F)F)OC)OC |
其他名称 | Act-078573 |
储存条件 | Store lyophilized at -20ºC, keep desiccated. |
Calculate the dilution required to prepare a stock solution. This equation is commonly abbreviated as: C1V1 = C2V2