AM095
目录号: A13981
LPA1 receptor 拮抗剂
AM095 是一种强效的 LPA1 受体拮抗剂,因为它能够抑制在过表达重组人类或小鼠 LPA1 的中国仓鼠卵巢(CHO)细胞膜上的 GTPγS 结合,其 IC50 值分别为 0.98 和 0.73 微米,并且没有表现出 LPA1 激动作用。
Discription | AM095 is a potent LPA1 receptor antagonist because it inhibited GTP??S binding to Chinese hamster ovary (CHO) cell membranes overexpressing recombinant human or mouse LPA1 with IC50 values of 0.98 and 0.73 μM, respectively, and exhibited no LPA1 agonism. |
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目录号 | A13981 |
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分子式 | C27H23N2NaO5 |
分子量 | 478.47 |
CAS号 | 1345614-59-6 |
SMILES | CC1=NOC(=C1NC(=O)O[C@H](C)C2=CC=CC=C2)C3=CC=C(C=C3)C4=CC=C(C=C4)CC(=O)[O-].[Na+] |
其他名称 | AM 095, AM-095 |
储存条件 | Store lyophilized at -20ºC, keep desiccated. |
Calculate the dilution required to prepare a stock solution. This equation is commonly abbreviated as: C1V1 = C2V2