AMG-1694
目录号: A21723
GK-GKRP disruptors
AMG-1694 是一种强效的葡萄糖激酶与葡萄糖激酶调节蛋白(GK-GKRP)解离剂,能促进 GK-GKRP 复合体的解离,其半抑制浓度(IC50)为 7 纳摩尔,间接增加了 GK 的酶活性。
Discription | AMG-1694 is a potent glucokinase?Cglucokinase regulatory protein (GK-GKRP) disruptors and promotes the dissociation of the GK-GKRP complex with an IC50 of 7 nM, indirectly increasing GK enzymatic activity. | |||||
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Cell Research |
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目录号 | A21723 |
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分子式 | C23H30F3N3O4S2 |
分子量 | 533.63 |
CAS号 | 1361217-07-3 |
SMILES | C[C@@](O)(C1=CC=C(N2[C@@H](CN3[C@@H](C)COCC3)CN(S(=O)(C4=CC=CS4)=O)CC2)C=C1)C(F)(F)F |
其他名称 | AMG1694, AMG 1694 |
储存条件 | Store lyophilized at -20ºC, keep desiccated. |
Calculate the dilution required to prepare a stock solution. This equation is commonly abbreviated as: C1V1 = C2V2