AMG9810
目录号: A19555
TRPV1 antagonist
AMG9810 是一种选择性和竞争性的范尼洛叶受体1(TRPV1)拮抗剂,其 IC50 值分别为人类和大鼠 TRPV1 的 24.5 和 85.6 nM。
Discription | AMG9810 is a selective and competitive vanilloid receptor 1 (TRPV1) antagonist with IC50 values of 24.5 and 85.6 nM for human and rat TRPV1, repectively. | |||||
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Cell Research |
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目录号 | A19555 |
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分子式 | C21H23NO3 |
分子量 | 337.41 |
CAS号 | 545395-94-6 |
SMILES | O=C(NC1=CC=C(OCCO2)C2=C1)/C=C/C3=CC=C(C(C)(C)C)C=C3 |
其他名称 | AMG-9810; AMG 9810 |
储存条件 | Store lyophilized at -20ºC, keep desiccated. |
In vitro | DMSO | 64 mg/mL (189.68 mM) | |
Water | Insoluble | ||
Ethanol | 24 mg/mL (71.13 mM) | ||
* <1 mg/ml means slightly soluble or insoluble. * Please note that Adooq tests the solubility of all compounds in-house, and the actual solubility may differ slightly from published values. This is normal and is due to slight batch-to-batch variations. |
Concentration / Solvent Volume / Mass | 1 mg | 5 mg | 10 mg |
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0.1 mM | 29.64 mL | 148.19 mL | 296.38 mL |
0.5 mM | 5.93 mL | 29.64 mL | 59.28 mL |
1 mM | 2.96 mL | 14.82 mL | 29.64 mL |
5 mM | 0.59 mL | 2.96 mL | 5.93 mL |
Calculate the dilution required to prepare a stock solution. This equation is commonly abbreviated as: C1V1 = C2V2