AMPK

Catalog No.Inhibitor Name AMPK
A13720Dorsomorphin 2HCl
**
A14312WZ4003
****
A11970Dorsomorphin
**
A16281HTH-01-015
***
A11071A 769662
*
A15815ETC-1002

Notes:
1.Hover mouse over " * " to view the IC50 value.(A few compounds have proven potency but without published IC50 data.)
2.For more details about the compound, click on the product name of your interest.
3.The higher the number of " * " is, the more potent the inhibitor or activator is.
4."" refers to compounds which do inhibitory effects on the related isoform, but without specific value.

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  1. WZ4003

    Catalog No. A14312
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    NUAK kinase 抑制剂
    WZ4003是一种高度特异性的NUAK激酶抑制剂,对于NUAK1和NUAK2的IC50为20 nM和100 nM。 了解更多
  2. HTH-01-015

    Catalog No. A16281
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    NUAK1 抑制剂
    HTH-01-015是NUAK1的有效和选择性抑制剂(IC50 = 100 nM),并且不影响包括其他AMPK家族成员在内的139种其他激酶的活性。 了解更多
  3. BML-275 (Dorsomorphin)

    Catalog No. A11970
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    AMPK 抑制剂
    BML-275 (Dorsomorphin)是一种可渗透细胞的吡唑并嘧啶化合物,显示为AMP激活的蛋白激酶(AMPK)和脂肪酸合酶抑制剂。 了解更多
  4. Dorsomorphin 2HCl

    Catalog No. A13720
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    BMP 抑制剂
    Dorsomorphin 2HCl (BML-275)是BMP信号传导的选择性小分子抑制剂,可促进胚胎干细胞的心肌发生。Dorsomorphin通过抑制骨形态发生蛋白信号转导逆转乳腺癌起始细胞的间质表型。 了解更多
  5. ETC-1002

    Catalog No. A15815
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    ACL 抑制剂 and AMPK 激活剂
    ETC-1002是一种新颖的,一流的可以降低LDL-C的小分子;肝AMP激活的蛋白激酶(AMPK)的激活剂;对肝ATP-柠檬酸裂解酶也具有有效的抑制活性(IC50 = 29 uM)。 了解更多

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