AMPK
Catalog No. | Inhibitor Name | AMPK |
---|---|---|
A13720 | Dorsomorphin 2HCl | ** |
A14312 | WZ4003 | **** |
A11970 | Dorsomorphin | ** |
A16281 | HTH-01-015 | *** |
A11071 | A 769662 | * |
A15815 | ETC-1002 |
Notes:
1.Hover mouse over " " to view the IC50 value.(A few compounds have proven potency but without published IC50 data.)
2.For more details about the compound, click on the product name of your interest.
3.The higher the number of " " is, the more potent the inhibitor or activator is.
4."" refers to compounds which do inhibitory effects on the related isoform, but without specific value.
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WZ4003
Catalog No. A14312 -
HTH-01-015
Catalog No. A16281 NUAK1 抑制剂HTH-01-015是NUAK1的有效和选择性抑制剂(IC50 = 100 nM),并且不影响包括其他AMPK家族成员在内的139种其他激酶的活性。 了解更多 -
BML-275 (Dorsomorphin)
Catalog No. A11970 AMPK 抑制剂BML-275 (Dorsomorphin)是一种可渗透细胞的吡唑并嘧啶化合物,显示为AMP激活的蛋白激酶(AMPK)和脂肪酸合酶抑制剂。 了解更多 -
Dorsomorphin 2HCl
Catalog No. A13720 BMP 抑制剂Dorsomorphin 2HCl (BML-275)是BMP信号传导的选择性小分子抑制剂,可促进胚胎干细胞的心肌发生。Dorsomorphin通过抑制骨形态发生蛋白信号转导逆转乳腺癌起始细胞的间质表型。 了解更多