AMY-101 TFA
目录号: A22779
AMY-101 TFA(Cp40 TFA),一种针对中心补体成分 C3 的肽类抑制剂(KD = 0.5 nM),能够抑制非人类灵长类动物(NHPs)中自然发生的牙周炎。AMY-101(Cp40)在COVID-19重症肺炎伴随系统性高炎症的模型中表现出良好的抗炎活性。
Discription | AMY-101 TFA (Cp40 TFA), a peptidic inhibitor of the central complement component C3 (KD = 0.5 nM), inhibits naturally occurring periodontitis in non-human primates (NHPs). AMY-101 (Cp40) exhibits a favorable anti-inflammatory activity in models with COVID-19 severe pneumonia with systemic hyper inflammation. |
---|
目录号 | A22779 |
---|---|
分子式 | C83H117N23O18S2.xC2HF3O2 |
CAS号 | 1789738-04-0 |
Sequence shortening | YICV-{Trp(Me)}-QDW-{Sar}-AHRC-{N(Me)Ile}-NH2 (Disulfide bridge:Cys3-Cys13) |
其他名称 | Cp40 TFA |
Calculate the dilution required to prepare a stock solution. This equation is commonly abbreviated as: C1V1 = C2V2