Anagliptin
目录号: A13529
DPP-4 抑制剂
Anagliptin 是一种强效且选择性的 DPP-4 抑制剂(IC50 = 3.8 nM);对 DPP-8 和 DPP-9 的抑制作用低于10倍。
Discription | Anagliptin is a potent and selective DPP-4 inhibitor(IC50= 3.8 nM); > 10 fold less potent for DPP-8 and DPP-9. | |||||
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Targets |
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Cell Research |
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目录号 | A13529 |
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分子式 | C19H25N7O2 |
分子量 | 383.45 |
CAS号 | 739366-20-2 |
SMILES | CC1=NN2C=C(C=NC2=C1)C(=O)NCC(C)(C)NCC(=O)N3CCC[C@H]3C#N |
其他名称 | SK-0403 |
储存条件 | Store lyophilized at -20ºC, keep desiccated. |
In vitro | DMSO | 74 mg/mL (192.98 mM) | |
Water | 19 mg/mL (49.54 mM) | ||
Ethanol | 74 mg/mL (192.98 mM) | ||
* <1 mg/ml means slightly soluble or insoluble. * Please note that Adooq tests the solubility of all compounds in-house, and the actual solubility may differ slightly from published values. This is normal and is due to slight batch-to-batch variations. |
Concentration / Solvent Volume / Mass | 1 mg | 5 mg | 10 mg |
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0.1 mM | 26.08 mL | 130.4 mL | 260.79 mL |
0.5 mM | 5.22 mL | 26.08 mL | 52.16 mL |
1 mM | 2.61 mL | 13.04 mL | 26.08 mL |
5 mM | 0.52 mL | 2.61 mL | 5.22 mL |
Calculate the dilution required to prepare a stock solution. This equation is commonly abbreviated as: C1V1 = C2V2