APG-115
目录号: A12575
MDM2 抑制剂
APG-115 (AA-115) 是一种口服活性的 MDM2 蛋白抑制剂,与 MDM2 蛋白 结合,其 IC50 和 Ki 值分别为 3.8 nM 和 1 nM。
Discription | APG-115 (AA-115) is an orally active MDM2 protein inhibitor binding to MDM2 protein with IC50 and Ki values of 3.8 nM and 1 nM, respectively. | |||||
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Cell Research |
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目录号 | A12575 |
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分子式 | C34H38Cl2FN3O4 |
分子量 | 642.59 |
CAS号 | 1818393-16-6 |
SMILES | O=C1NC2=CC(Cl)=CC=C2[C@]13C4(CCCCC4)N(CC)[C@@H](C(NC56CCC(CC6)(C(O)=O)CC5)=O)[C@@H]3C7=C(C(Cl)=CC=C7)F |
其他名称 | APG115, APG 115 |
储存条件 | Store lyophilized at -20ºC, keep desiccated. |
Calculate the dilution required to prepare a stock solution. This equation is commonly abbreviated as: C1V1 = C2V2