Argatroban

Name: Argatroban
SKU: A11774

目录号: A11774

Thrombin 抑制剂

Argatroban Chemical Structure

CAS NO. 74863-84-6

Argatroban是一种抗凝剂，是一种小分子直接凝血酶抑制剂，Ki值范围为5 nM-39 nM。

库存：现货

规格	价格	数量
10 mg	￥ 490.00
25 mg	￥ 1,050.00
50 mg	￥ 1,540.00
100 mg	￥ 2,660.00

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Argatroban是一种抗凝剂，是一种小分子直接凝血酶抑制剂，Ki值范围为5 nM-39 nM。

靶点信息

Thrombin
5-39 nM(Ki)

溶解度 *

In vitro (25°C)	DMSO	8 mg/mL (15.72 mM)
	Water	Insoluble
	Ethanol	5 mg/mL (9.83 mM)
In vivo	2% DMSO+40% PEG 300+2% Tween 80+ddH2O	4 mg/mL
* <1 mg/ml means slightly soluble or insoluble. * Please note that Adooq tests the solubility of all compounds in-house, and the actual solubility may differ slightly from published values. This is normal and is due to slight batch-to-batch variations.

制备储备液

Concentration / Solvent Volume / Mass	1 mg	5 mg	10 mg
0.1 mM	19.66 mL	98.31 mL	196.62 mL
0.5 mM	3.93 mL	19.66 mL	39.32 mL
1 mM	1.97 mL	9.83 mL	19.66 mL
5 mM	0.39 mL	1.97 mL	3.93 mL

*The above data is based on the productmolecular weight 508.6 . Batch specific molecular weights may vary from batch to batch due to solvent of hydration, which will affect the solvent volumes required to prepare stock solutions.

化学数据

目录号	A11774
作用机制	Inhibitor (抑制剂)
M. Wt	508.6
Formula	C23H36N6O5S
Purity	>99%
Storage	Store lyophilized at -20ºC, keep desiccated. In lyophilized form, the chemical is stable for 36 months. In solution, store at -20ºC and use within 3 months to prevent loss of potency. Aliquot to avoid multiple freeze/thaw cycles.
CAS No.	74863-84-6
SMILES	C[C@@H]1CCN([C@H](C1)C(=O)O)C(=O)[C@H](CCCN=C(N)N)NS(=O)(=O)C2=CC=CC3=C2NCC(C3)C