ASP4132
目录号: A22339
AMPK activator
ASP4132 是一种口服活性强、效力高的 AMPK 激活剂,其 EC50 为 18 nM。ASP4132 具有抗癌活性,并能在乳腺癌异种移植小鼠模型中引起肿瘤退缩。
Discription | ASP4132 is an orally active, potent AMPK activator with an EC50 of 18 nM. ASP4132 has anti-cancer activity and makes tumor regression in breast cancer xenograft mouse models. | |||||
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Cell Research |
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目录号 | A22339 |
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分子式 | C46H51F3N6O8S2 |
分子量 | 937.06 |
CAS号 | 1640294-30-9 |
SMILES | O=C(C1=NC2=CC=C(C3CCN(CC4=CC=C(OC)N=C4)CC3)C=C2N1)N5CCN(CC6=CC=C(C(F)(F)F)C=C6)CC5.O=S(C7=CC=C(C)C=C7)(O)=O.O=S(C8=CC=C(C)C=C8)(O)=O |
其他名称 | ASP-4132,ASP 4132 |
储存条件 | Store lyophilized at -20ºC, keep desiccated. |
Calculate the dilution required to prepare a stock solution. This equation is commonly abbreviated as: C1V1 = C2V2