Balovaptan
目录号: A19373
hV1a receptor antagonist
Balovaptan (RG7314) 是一种高效且选择性的能穿透大脑的抗利尿激素1a(hV1a)受体拮抗剂,对人类(hV1a)和小鼠(mV1a)受体的Kis分别为1 nM和39 nM,用于自闭症的研究。
Discription | Balovaptan (RG7314) is a highly potent and selective brain-penetrant vasopressin 1a (hV1a) receptor antagonist, with Kis of 1 and 39 nM for human (hV1a) and mouse (mV1a) receptors, and is used for the research of autism. |
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目录号 | A19373 |
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分子式 | C22H24ClN5O |
分子量 | 409.91 |
CAS号 | 1228088-30-9 |
SMILES | CN1CC2=NN=C([C@H]3CC[C@H](OC4=NC=CC=C4)CC3)[N@]2[C@]5=CC=C(Cl)C=C5C1 |
其他名称 | RG7314, RG-7314, RG 7314 |
储存条件 | Store lyophilized at -20ºC, keep desiccated. |
Calculate the dilution required to prepare a stock solution. This equation is commonly abbreviated as: C1V1 = C2V2