BDP5290
目录号: A16966
ROCK and MRCK 抑制剂
BDP5290 是一种强效的 ROCK 和 MRCK 抑制剂,其半抑制浓度(IC50)分别为 ROCK1 5 nM、ROCK2 50 nM、MRCKα 10 nM 和 MRCKβ 100 nM。
Discription | BDP5290 is a potent inhibitor of both ROCK and MRCK with IC50s of 5 nM, 50 nM, 10 nM and 100 nM for ROCK1, ROCK2, MRCKα and MRCKβ, respectively. | ||
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目录号 | A16966 |
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分子式 | C17H18ClN7O |
分子量 | 371.82 |
CAS号 | 1817698-21-7 |
SMILES | ClC(C(C(NC1=CNN=C1C2=NC=CC=C2)=O)=N3)=CN3C4CCNCC4 |
其他名称 | BDP 5290, BDP-5290 |
储存条件 | Store lyophilized at -20ºC, keep desiccated. |
Calculate the dilution required to prepare a stock solution. This equation is commonly abbreviated as: C1V1 = C2V2