BI-3802
目录号: A19733
BI-3802 是一种高效的 BCL6 降解剂,能够抑制 BCL6 的 BTB 域,IC50 值约为 3 nM;BI-3802 具有抗肿瘤活性。
Discription | BI-3802 is a highly potent BCL6 degrader, inhibiting the BTB domain of BCL6, with an IC50 of ??3 nM; BI-3802 has antitumor activity. |
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目录号 | A19733 |
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分子式 | C24H29ClN6O3 |
分子量 | 484.98 |
CAS号 | 2166387-65-9 |
SMILES | ClC1=CN=C(N2C[C@H](C)C[C@H](C)C2)N=C1NC3=CC(C=C(OCC(NC)=O)C(N4C)=O)=C4C=C3 |
其他名称 | U52; U-52; U 52; BI-3802; BI 3802; BI3802 |
储存条件 | Store lyophilized at -20ºC, keep desiccated. |
In vitro | DMSO | 3 mg/mL (6.18 mM) | |
Water | Insoluble | ||
Ethanol | Insoluble | ||
* <1 mg/ml means slightly soluble or insoluble. * Please note that Adooq tests the solubility of all compounds in-house, and the actual solubility may differ slightly from published values. This is normal and is due to slight batch-to-batch variations. |
Concentration / Solvent Volume / Mass | 1 mg | 5 mg | 10 mg |
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0.1 mM | 20.62 mL | 103.1 mL | 206.19 mL |
0.5 mM | 4.12 mL | 20.62 mL | 41.24 mL |
1 mM | 2.06 mL | 10.31 mL | 20.62 mL |
5 mM | 0.41 mL | 2.06 mL | 4.12 mL |
Calculate the dilution required to prepare a stock solution. This equation is commonly abbreviated as: C1V1 = C2V2