BI-9564
目录号: A16196
BRD7/9 抑制剂
BI-9564 是一种强效且选择性的 BRD9 和 BRD7 溴结构域抑制剂(Kds 分别为 14.1 和 239 nM;IC50s 分别为 75 nM 和 3.4 uM)。
Discription | BI-9564 is a potent and selective inhibitor of BRD9 and BRD7 bromodomains (Kds = 14.1 and 239 nM; IC50s = 75 nM and 3.4 uM, respectively). | |||||
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Cell Research |
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目录号 | A16196 |
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分子式 | C20H23N3O3 |
分子量 | 353.41 |
CAS号 | 1883429-22-8 |
SMILES | O=C1N(C)C=C(C2=CC(OC)=C(CN(C)C)C=C2OC)C3=CC=NC=C13 |
其他名称 | BI 9564, BI9564 |
储存条件 | Store lyophilized at -20ºC, keep desiccated. |
In vitro | DMSO | 3 mg/mL (8.48 mM) | |
Water | Insoluble | ||
Ethanol | 15 mg/mL (42.44 mM) | ||
* <1 mg/ml means slightly soluble or insoluble. * Please note that Adooq tests the solubility of all compounds in-house, and the actual solubility may differ slightly from published values. This is normal and is due to slight batch-to-batch variations. |
Concentration / Solvent Volume / Mass | 1 mg | 5 mg | 10 mg |
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0.1 mM | 28.3 mL | 141.48 mL | 282.96 mL |
0.5 mM | 5.66 mL | 28.3 mL | 56.59 mL |
1 mM | 2.83 mL | 14.15 mL | 28.3 mL |
5 mM | 0.57 mL | 2.83 mL | 5.66 mL |
Calculate the dilution required to prepare a stock solution. This equation is commonly abbreviated as: C1V1 = C2V2