BMS-1166 hydrochloride
目录号: A21481
PD-1/PD-L1 interaction 抑制剂
BMS-1166 盐酸盐是一种强效的 PD-1/PD-L1 互作抑制剂,其 IC50 为 1.4 nM。BMS-1166 对 PD-1/PD-L1 免疫检查点在 T 细胞激活上的抑制效果具有拮抗作用。
Discription | BMS-1166 hydrochloride is a potent PD-1/PD-L1 interaction inhibitor with an IC50 of 1.4 nM. BMS-1166 antagonizes the inhibitory effect of PD-1/PD-L1 immune checkpoint on T cell activation. |
---|
目录号 | A21481 |
---|---|
分子式 | C36H34Cl2N2O7 |
分子量 | 677.57 |
CAS号 | 2113650-05-6 |
SMILES | O=C(O)[C@@H]1N(CC2=CC(Cl)=C(OCC3=CC=CC(C4=CC=C(OCCO5)C5=C4)=C3C)C=C2OCC6=CC=CC(C#N)=C6)C[C@H](O)C1.Cl |
其他名称 | BMS 1166 Hydrochloride; BMS1166 Hydrochloride; BMS-1166 HCl; BMS 1166 HCl; BMS1166 HCl |
储存条件 | Store lyophilized at -20ºC, keep desiccated. |
Calculate the dilution required to prepare a stock solution. This equation is commonly abbreviated as: C1V1 = C2V2