BMS-819881
目录号: A21500
MCHR1 antagonist
BMS-819881 是一种黑色素集中激素受体1(MCHR1)拮抗剂,其与大鼠MCHR1的结合Ki值为7 nM。BMS-819881 对CYP3A4活性也具有选择性和强效性,EC50值为13 μM。
Discription | BMS-819881 is a melaninconcentrating hormone receptor 1 (MCHR1) antagonist, which binds rat MCHR1 with a Ki of 7 nM. BMS-819881 also is selective and potent for CYP3A4 activity with an EC50 of 13 μM. | ||
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目录号 | A21500 |
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分子式 | C24H21ClN2O4S |
分子量 | 468.95 |
CAS号 | 1197420-05-5 |
SMILES | ClC1=CC=C(C2=CC(N=CN(C3=CC(OC)=C(OC[C@H](O)C4CC4)C=C3)C5=O)=C5S2)C=C1 |
其他名称 | BMS 819881; BMS819881 |
储存条件 | Store lyophilized at -20ºC, keep desiccated. |
Calculate the dilution required to prepare a stock solution. This equation is commonly abbreviated as: C1V1 = C2V2