Brompheniramine
目录号: A11699
溴苯那敏是一种第一代抗组胺药。溴苯那敏的作用机制是作为组胺H1受体的拮抗剂。它还具有中等效力的抗胆碱能作用,并可能是与二苯海拉明等常见抗组胺药类似的抗毒蕈碱作用剂。
Discription | Brompheniramine is a first-generation antihistamine. Brompheniramine works by acting as an antagonist of histamine H1 receptors. It also functions as a moderately effective anticholinergic agent, and is likely an antimuscarinic agent similar to other common antihistamines such as diphenhydramine. | ||
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目录号 | A11699 |
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分子式 | C16H19BrN2.C4H4O4 |
分子量 | 435.31 |
CAS号 | 980-71-2 |
SMILES | CN(C)CCC(C1=CC=C(C=C1)Br)C2=CC=CC=N2.C(=C\C(=O)O)\C(=O)O |
储存条件 | Store lyophilized at -20ºC, keep desiccated. |
In vitro | DMSO | 78 mg/mL (179.18 mM) | |
Water | Warmed: 41 mg/mL (94.18 mM) | ||
Ethanol | 16 mg/mL (36.75 mM) | ||
* <1 mg/ml means slightly soluble or insoluble. * Please note that Adooq tests the solubility of all compounds in-house, and the actual solubility may differ slightly from published values. This is normal and is due to slight batch-to-batch variations. |
Concentration / Solvent Volume / Mass | 1 mg | 5 mg | 10 mg |
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0.1 mM | 22.97 mL | 114.86 mL | 229.72 mL |
0.5 mM | 4.59 mL | 22.97 mL | 45.94 mL |
1 mM | 2.3 mL | 11.49 mL | 22.97 mL |
5 mM | 0.46 mL | 2.3 mL | 4.59 mL |
Calculate the dilution required to prepare a stock solution. This equation is commonly abbreviated as: C1V1 = C2V2