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￥ 0.00 CaMK
| Catalog No. | Inhibitor Name | CaMKII | CaMKIII | CaMKKα | CaMKKβ | Other |
|---|---|---|---|---|---|---|
| A14307 | NH125 | **** | PKC,PKA | |||
| A11473 | KN-62 | ** | ||||
| A14288 | KN-93 Phosphate | *** | ||||
| A16345 | STO-609 acetate | *** | **** | |||
| A13804 | CID 755673 | * | PKD1, PKD2, PKD3, PKC, CAK, PLK1, Akt | |||
| A13447 | A-484954 | *** |
Notes:
1.Hover mouse over "" to view the IC50 value.(A few compounds have proven potency but without published IC50 data.)
2.For more details about the compound, click on the product name of your interest.
3.The higher the number of "" is, the more potent the inhibitor or activator is.
4."" refers to compounds which do inhibitory effects on the related isoform, but without specific value.
17 个项目
每页
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CaMKII-IN-1
Catalog No. A21034 CaMKII inhibitorCaMKII-IN-1 is a potent and highly selective CaMKII inhibitor with IC50 of 63 nM. 了解更多 -
STO-609 acetate
Catalog No. A16345 -
CRT-0066101
Catalog No. A16318 PKD 抑制剂CRT-0066101是有效，选择性的蛋白激酶D（PKD）抑制剂；抑制所有PKD同工型（PKD1，PKD3和PKD2的IC50值分别为1、2和2.5 nM）。 了解更多 -
CID 797718
Catalog No. A13809 PKD1 抑制剂CID797718是CID755673（Adooq目录号A13804）的结构类似物。它是效力降低10倍的PKD1抑制剂，IC50值为7.0+/-0.8 uM。 了解更多 -
KN-92 phosphate
Catalog No. A15139 CaMKII 抑制剂KN-92 phosphate是KN-93的非活性衍生物。KN-93是Ca2+/钙调蛋白依赖性激酶II（CaMKII）的选择性抑制剂，竞争性阻断CaM与激酶的结合（Ki = 370 nM）。 了解更多 -
KN-92 hydrochloride
Catalog No. A15138 -
A-484954
Catalog No. A13447 -
K252a
Catalog No. A13897 -
KN-93 Phosphate
Catalog No. A14288 CaMKII 抑制剂KN-93 Phosphate是一种有效且特异性的Ca2+/钙调蛋白依赖性蛋白激酶II（CaMKII）抑制剂，Ki为0.37μM，对APK，PKC，MLCK或Ca2+-PDE活性无明显抑制作用。 了解更多 -
CID 755673
Catalog No. A13804 PKD 抑制剂CID755673是一种具有细胞活性的泛PKD1/2/3抑制剂，IC50值分别为180 nM，280nM，以及227 nM。 了解更多 -
Phenoxybenzamine hydrochloride
Catalog No. A10719 α-adrenergic (AR) 拮抗剂/CaM 抑制剂Phenoxybenzamine hydrochloride是一种细胞可渗透的，非特异性的，不可逆的α-肾上腺素（AR）拮抗剂，也可作为CaM抑制剂。 了解更多 -
kb NB 142-70
Catalog No. A12423 -
CID 2011756
Catalog No. A12416 -
KN-62
Catalog No. A11473
17 个项目
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- Inhibitor (抑制剂) (17)
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