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Cannabinoid Receptors

26 个项目

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  1. Taranabant ((1R,2R)stereoisomer)
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    Taranabant ((1R,2R)stereoisomer)

    Catalog No. A21705
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    CB1 receptor inverse agonist
    Taranabant (1R,2R)stereoisomer is the R-enantiomer of Taranabant. Taranabant is a highly potent and selective cannabinoid 1 (CB1) receptor inverse agonist. 了解更多
  2. Taranabant racemate
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    Taranabant racemate

    Catalog No. A21699
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    CB1 antagonist/inverse agonist
    Taranabant racemate is an antagonist and/or inverse agonist of the Cannabinoid-1 (CB1) receptor extracted from patent WO 2004048317 A1. 了解更多
  3. (±)-Ibipinabant
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    (±)-Ibipinabant

    Catalog No. A21439
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    CB-1 receptor antagonist
    (±)-Ibipinabant ((±)-SLV319) is the racemate of SLV319. (±)-Ibipinabant ((±)-SLV319) is a potent and selective cannabinoid-1 (CB-1) receptor antagonist with an IC50 of 22 nM. 了解更多
  4. JD-5037
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    JD-5037

    Catalog No. A20837
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    CB1R antagonist
    JD-5037 is a novel, peripherally restricted CB1R antagonist with an IC50 of 1.5 nM. 了解更多
  5. Taranabant
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    Taranabant

    Catalog No. A11578
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    CB1 receptor inverse agonist
    Taranabant is a highly potent and selective cannabinoid 1 (CB1) receptor inverse agonist that inhibits the binding and functional activity of various agonists, with a binding Ki of 0.13 nM for the human CB1R in vitro. 了解更多
  6. CB2R-IN-1
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    CB2R-IN-1

    Catalog No. A12306
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    cannabinoid CB2 receptor inverse agonist
    CB2R-IN-1 is a potent cannabinoid CB2 receptor inverse agonist with a Ki of 0.9 nM. 了解更多
  7. CB1 antagonist 2
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    CB1 antagonist 2

    Catalog No. A18810
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    CB1 antagonist
    CB1 antagonist 2 is caimabinoid 1 (CB1) antagonist extracted from patent WO2016184310A1, compound 3, inhibits CB1 in vivo with an IC50 of 25.5 nM. 了解更多
  8. SR 144528
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    SR 144528

    Catalog No. A12376
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    CB2 inverse 激动剂
    SR 144528是一种选择性的外周大麻素受体反向激动剂，对大鼠脾脏和人重组CB2受体的Ki值为0.6 nM，对大鼠脑和人重组CB1受体的Ki值为400 nM。 了解更多
  9. GNE-049
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    GNE-049

    Catalog No. A20206
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    CBP inhibitor
    GNE-049 is a highly potent and selective CBP inhibitor with an IC50 of 1.1 nM in TR-FRET assay. GNE-049 also inhibits BRET and BRD4(1) with IC50s of 12 nM and 4200 nM, respectively. 了解更多
  10. VCE-004.8
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    VCE-004.8

    Catalog No. A18549
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    PPARγ and CB2 receptor dual agonist
    VCE-004.8, a semi-synthetic multitarget cannabinoquinoid, is a specific PPARγ and CB2 receptor dual agonist with potent anti-inflammatory activity. 了解更多
  11. Rimonabant hydrochloride
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    Rimonabant hydrochloride

    Catalog No. A11548
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    CB1 receptor inverse 激动剂
    Rimonabant hydrochloride是CB1受体反向激动剂。 了解更多
  12. AM1241
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    AM1241

    Catalog No. A16397
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    CB2 receptor 激动剂
    AM1241是选择性的大麻素CB2受体激动剂，Ki为3.4 nM，相对于CB1受体具有82倍的选择性。 了解更多
  13. Bay 59-3074
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    Bay 59-3074

    Catalog No. A16328
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    CB1/CB2 receptor 激动剂
    Bay 59-3074是一种新型的选择性CB1/CB2受体部分激动剂，对人CB1和CB2受体的Ki值分别为48.3和45.5 nM。 了解更多
  14. AM630
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    AM630

    Catalog No. A14993
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    CB2 拮抗剂
    AM630是一种选择性CB2拮抗剂，Ki为31.2 nM，选择性是CB1受体的150倍以上。 了解更多
  15. Otenabant
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    Otenabant

    Catalog No. A15200
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    CB1 receptor 拮抗剂
    Otenabant是最近发现的选择性，高亲和力，竞争性CB1受体拮抗剂，Ki为0.7 nM。 了解更多
  16. Tedalinab
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    Tedalinab

    Catalog No. A14189
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    CB2 receptor 激动剂
    Tedalinab (GRC-10693)是开发用于治疗骨关节炎和神经性疼痛的药物，它可作为有效的选择性大麻素CB2受体激动剂。与相关的CB1受体相比，它对CB2的选择性为4700x，具有很高的口服生物利用度，并在早期临床试验中显示出令人鼓舞的安全性结果以及有效的镇痛和抗炎作用。 了解更多
  17. AM 2201
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    AM 2201

    Catalog No. A14174
    Cannabinoid 抑制剂
    AM2201是有效的合成大麻素（CB），对于CB1和CB2受体的Ki值分别为1.0和2.6 nM。 了解更多
  18. AM251
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    AM251

    Catalog No. A12914
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    CB1 receptor 拮抗剂
    AM251是有效的CB1受体拮抗剂（IC50 = 8 nM，Ki = 7.49 nM），其选择性是CB2受体的306倍。 了解更多
  19. Org 27569
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    Org 27569

    Catalog No. A11513
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    CB1 modulator?
    Org 27569是一种强效CB1受体变构调节剂(PEC50 = 8.24)。 了解更多
  20. Rimonabant (SR141716)
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    Rimonabant (SR141716)

    Catalog No. A11547
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    Rimonabant是CB1的选择性拮抗剂，在hCB1转染的HEK 293膜中的IC50为13.6 nM，EC50为17.3 nM。 了解更多
  21. GW842166X
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    GW842166X

    Catalog No. A11253
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    CB2 receptor 激动剂
    GW842166X是一种选择性的非大麻类CB2受体激动剂，EC50为63 nM，对CB1受体没有显著的活性。 了解更多
  22. CP 945598 HCl (Otenabant HCl)
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    CP 945598 HCl (Otenabant HCl)

    Catalog No. A11942
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    CB1 拮抗剂
    CP 945598 HCl (Otenabant HCl)是一种有效且高度选择性的CB1拮抗剂。 了解更多
  23. MDA 19
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    MDA 19

    Catalog No. A11939
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    CB2 激动剂
    MDA 19是CB2的有效选择性激动剂，对精神活性CB1受体具有合理的选择性。 了解更多
  24. BML-190
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    BML-190

    Catalog No. A11938
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    CB2 receptor ligand
    BML-190是CB2受体的选择性反向激动剂。 了解更多
  25. WIN 55,212-2 mesylate
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    WIN 55,212-2 mesylate

    Catalog No. A11932
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    CB receptor 激动剂
    WIN 55,212-2 mesylate是一种有效的cannabinoid receptor激动剂，在神经性疼痛的大鼠模型中具有有效的镇痛作用。它通过受体介导的信号激活p42和p44 MAP激酶。 了解更多
  26. UR-144
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    UR-144

    Catalog No. A11096
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    UR-144是有效的合成大麻素（CB），其优先结合周围的CB2受体（Ki = 1.8 nM）超过中央CB1受体（Ki = 150 nM）。 了解更多

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  1. Inhibitor (抑制剂) (2)
  2. Agonist (激动剂) (12)
  3. Antagonist (拮抗剂) (8)
  4. Modulator (调节剂) (1)
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