CC-90003
目录号: A16837
ERK1/2 抑制剂
CC-90003 是一种不可逆的 ERK1/2 抑制剂,其 IC50 在 10-20 nM 范围内,并在 258-激酶生化测定中显示出良好的激酶选择性。
Discription | CC-90003 is an irreversible inhibitor of ERK1/2 with IC50s in the 10-20 nM range and shows good kinase selectivity in a 258-kinase biochemical assay. | ||
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目录号 | A16837 |
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分子式 | C22H21F3N6O2 |
分子量 | 458.44 |
CAS号 | 1621999-82-3 |
SMILES | C=CC(NC1=CC(C)=CC=C1NC2=NC(NC3=CC(OC)=NC=C3C)=NC=C2C(F)(F)F)=O |
其他名称 | CC 90003, CC90003 |
储存条件 | Store lyophilized at -20ºC, keep desiccated. |
In vitro | DMSO | 78 mg/mL (170.14 mM) | |
Water | Insoluble | ||
Ethanol | Insoluble | ||
* <1 mg/ml means slightly soluble or insoluble. * Please note that Adooq tests the solubility of all compounds in-house, and the actual solubility may differ slightly from published values. This is normal and is due to slight batch-to-batch variations. |
Concentration / Solvent Volume / Mass | 1 mg | 5 mg | 10 mg |
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0.1 mM | 21.81 mL | 109.07 mL | 218.13 mL |
0.5 mM | 4.36 mL | 21.81 mL | 43.63 mL |
1 mM | 2.18 mL | 10.91 mL | 21.81 mL |
5 mM | 0.44 mL | 2.18 mL | 4.36 mL |
Calculate the dilution required to prepare a stock solution. This equation is commonly abbreviated as: C1V1 = C2V2