Celastrol

Name: Celastrol
SKU: A10192

目录号: A10192

Product Citations (2)

Celastrol Chemical Structure

CAS NO. 34157-83-0

Celastrol是一种有效的蛋白酶抑制剂，有效且优先抑制胰凝乳蛋白酶样的纯化的20S proteasome的活性，IC50为2.5 μM。

库存：现货

规格	价格	数量
10 mg	￥ 350.00
25 mg	￥ 630.00
50 mg	￥ 910.00
100 mg	￥ 1,225.00

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生物活性

Celastrol是一种有效的蛋白酶抑制剂，有效且优先抑制胰凝乳蛋白酶样的纯化的20S proteasome的活性，IC50为2.5 μM。

靶点信息

20S proteasome	20S proteasome
N/A	2.5 μM

溶解度 *

In vitro	DMSO	82 mg/mL (181.97 mM)
	Water	Insoluble
	Ethanol	Insoluble
* <1 mg/ml means slightly soluble or insoluble. * Please note that Adooq tests the solubility of all compounds in-house, and the actual solubility may differ slightly from published values. This is normal and is due to slight batch-to-batch variations.

制备储备液

Concentration / Solvent Volume / Mass	1 mg	5 mg	10 mg
0.1 mM	22.19 mL	110.96 mL	221.93 mL
0.5 mM	4.44 mL	22.19 mL	44.39 mL
1 mM	2.22 mL	11.1 mL	22.19 mL
5 mM	0.44 mL	2.22 mL	4.44 mL

*The above data is based on the productmolecular weight 450.6 . Batch specific molecular weights may vary from batch to batch due to solvent of hydration, which will affect the solvent volumes required to prepare stock solutions.

化学数据

目录号	A10192
M. Wt	450.6
Formula	C29H38O4
Purity	>99%
Storage	Store lyophilized at -20ºC, keep desiccated. In lyophilized form, the chemical is stable for 36 months. In solution, store at -20ºC and use within 3 months to prevent loss of potency. Aliquot to avoid multiple freeze/thaw cycles.
CAS No.	34157-83-0
SMILES	CC1=C(C(=O)C=C2C1=CC=C3[C@]2(CC[C@@]4([C@@]3(CC[C@@]5([C@H]4C[C@](CC5)(C)C(=O)O)C)C)C)C)O