Cenicriviroc
目录号: A13643
CCR2/CCR5 抑制剂
Cenicriviroc 是一种用于治疗 HIV 感染的实验性药物候选。Cenicriviroc 是 CCR2 和 CCR5 受体的抑制剂,使其能够作为进入抑制剂,阻止病毒进入人体细胞。
Discription | Cenicriviroc is an experimental drug candidate for the treatment of HIV infection.Cenicriviroc is an inhibitor of CCR2 and CCR5 receptors, allowing it to function as an entry inhibitor which prevents the virus from entering into a human cell. | ||
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Targets |
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目录号 | A13643 |
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分子式 | C41H52N4O4S |
分子量 | 696.94 |
CAS号 | 497223-25-3 |
SMILES | CCCCOCCOC1=CC=C(C=C1)C2=CC/3=C(C=C2)N(CCC/C(=C3)/C(=O)NC4=CC=C(C=C4)[S@@](=O)CC5=CN=CN5CCC)CC(C)C |
其他名称 | TAK-652, TBR-652 |
储存条件 | Store lyophilized at -20ºC, keep desiccated. |
In vitro | DMSO | 94 mg/mL (134.87 mM) | |
Water | Insoluble | ||
Ethanol | 94 mg/mL (134.87 mM) | ||
* <1 mg/ml means slightly soluble or insoluble. * Please note that Adooq tests the solubility of all compounds in-house, and the actual solubility may differ slightly from published values. This is normal and is due to slight batch-to-batch variations. |
Concentration / Solvent Volume / Mass | 1 mg | 5 mg | 10 mg |
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0.1 mM | 14.35 mL | 71.74 mL | 143.48 mL |
0.5 mM | 2.87 mL | 14.35 mL | 28.7 mL |
1 mM | 1.43 mL | 7.17 mL | 14.35 mL |
5 mM | 0.29 mL | 1.43 mL | 2.87 mL |
Calculate the dilution required to prepare a stock solution. This equation is commonly abbreviated as: C1V1 = C2V2