CEP-37440
目录号: A15543
FAK/ALK 抑制剂
CEP-37440 是一种新型的高效选择性 双重 FAK/ALK 抑制剂,其 IC50 值分别为 2.3 nM(FAK)和 120 nM(ALK 细胞 IC50 在 75% 人血浆中)。
Discription | CEP-37440 is a novel potent and selective Dual FAK/ALK inhibitor with IC50 s of 2.3 nM (FAK) and 120 nM(ALK cellular IC50 in 75% human plasma). |
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目录号 | A15543 |
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分子式 | C30H38ClN7O3 |
分子量 | 580.12 |
CAS号 | 1391712-60-9 |
SMILES | CNC(=O)C1=CC=CC=C1NC2=NC(=NC=C2Cl)NC3=C(C4=C(CC(CCC4)N5CCN(CC5)CCO)C=C3)OC |
其他名称 | CEP37440, CEP 37440 |
储存条件 | Store lyophilized at -20ºC, keep desiccated. |
Calculate the dilution required to prepare a stock solution. This equation is commonly abbreviated as: C1V1 = C2V2