CGP71683 hydrochloride
目录号: A19844
neuropeptide Y5 receptor antagonist
CGP71683 盐酸盐是一种竞争性神经肽Y5受体拮抗剂,具有 1.3 nM 的 Ki 值,在 Y1 受体(Ki 值 >4000 nM)和 Y2 受体(Ki 值 200 nM)上没有明显活性。
Discription | CGP71683 hydrochloride is a competitive neuropeptide Y5 receptor antagonist with a Ki of 1.3 nM, and shows no obvious activity at Y1 receptor (Ki, >4000 nM) and Y2 receptor (Ki, 200 nM) in cell membranes. |
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目录号 | A19844 |
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分子式 | C26H30ClN5O2S |
分子量 | 512.07 |
CAS号 | 192322-50-2 |
SMILES | O=S(C1=C2C=CC=CC2=CC=C1)(NC[C@H]3CC[C@H](CNC4=NC(N)=C5C=CC=CC5=N4)CC3)=O.Cl |
其他名称 | CGP 71683A, CGP-71683A, CGP71683A; CGP-71683, CGP 71683 |
储存条件 | Store lyophilized at -20ºC, keep desiccated. |
In vitro | DMSO | 88 mg/mL (171.85 mM) | |
Water | Insoluble | ||
Ethanol | Insoluble | ||
* <1 mg/ml means slightly soluble or insoluble. * Please note that Adooq tests the solubility of all compounds in-house, and the actual solubility may differ slightly from published values. This is normal and is due to slight batch-to-batch variations. |
Concentration / Solvent Volume / Mass | 1 mg | 5 mg | 10 mg |
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0.1 mM | 19.53 mL | 97.64 mL | 195.29 mL |
0.5 mM | 3.91 mL | 19.53 mL | 39.06 mL |
1 mM | 1.95 mL | 9.76 mL | 19.53 mL |
5 mM | 0.39 mL | 1.95 mL | 3.91 mL |
Calculate the dilution required to prepare a stock solution. This equation is commonly abbreviated as: C1V1 = C2V2