微信关注
Total item
Cart Subtotal
￥ 0.00 产品详情
CH5132799是一种新型的I类PI3K抑制剂，尤其对PI3Kα (IC (50) = 0.014μM) 表现出很强的抑制活性。
Targets
| Target | Value |
|---|---|
| PI3Kα | IC50: 14nM |
| PI3Kγ | IC50: 36nM |
| PI3Kβ | IC50: 0.12μM |
| PI3Kδ | IC50: 0.50μM |
| mTOR | IC50: 1.6μM |
| C2β | IC50: 5.3μM |
| C2α | IC50: >10μM |
| Vps34 | IC50: >10μM |
| In vitro (25°C) | DMSO | 12 mg/mL (31.79 mM) | |
| Water | Insoluble | ||
| Ethanol | Insoluble | ||
| In vivo | 1% DMSO+30% polyethylene glycol+1% Tween 80 | 28 mg/mL | |
|
* <1 mg/ml means slightly soluble or insoluble. * Please note that Adooq tests the solubility of all compounds in-house, and the actual solubility may differ slightly from published values. This is normal and is due to slight batch-to-batch variations. |
|||
| Concentration / Solvent Volume / Mass | 1 mg | 5 mg | 10 mg |
|---|---|---|---|
| 0.1 mM | 26.5 mL | 132.48 mL | 264.96 mL |
| 0.5 mM | 5.3 mL | 26.5 mL | 52.99 mL |
| 1 mM | 2.65 mL | 13.25 mL | 26.5 mL |
| 5 mM | 0.53 mL | 2.65 mL | 5.3 mL |
*The above data is based on the productmolecular weight 377.42. Batch specific molecular weights may vary from batch to batch due to solvent of hydration, which will affect the solvent volumes required to prepare stock solutions.
| 目录号 | A11169 |
|---|---|
| 作用机制 | Inhibitor (抑制剂) |
| M. Wt | 377.42 |
| Formula | C15H19N7O3S |
| Purity | >99% |
| Storage | Store lyophilized at -20ºC, keep desiccated. |
| CAS No. | 1007207-67-1 |
| Synonyms | CH-5132799 |
| SMILES | CS(=O)(=O)N1CCC2=C(N=C(N=C21)N3CCOCC3)C4=CN=C(N=C4)N |
产品标签
Product Questions
Product Questions
No Questions
Keywords:购买 CH5132799 | CH5132799 供应商 | 订购 CH5132799 | CH5132799 价格 | CH5132799 生产商 | 订单 CH5132799 | CH5132799 代理商 | 购买 1007207-67-1| 1007207-67-1 供应商 | 订购 1007207-67-1 | 1007207-67-1 价格 | 1007207-67-1 生产商 | 订单 1007207-67-1 | 1007207-67-1 代理商|buy CH5132799 | CH5132799 Supplier | purchase CH5132799 | CH5132799 cost | CH5132799 manufacturer | order CH5132799 | CH5132799 distributor | buy 1007207-67-1| 1007207-67-1 Supplier | purchase 1007207-67-1 | 1007207-67-1 cost | 1007207-67-1 manufacturer | order 1007207-67-1 | 1007207-67-1 distributor