CI 972
目录号: A18598
PNP 抑制剂
CI 972 是一种强效的、口服活性的、竞争性的嘌呤核苷磷酸化酶(PNP)抑制剂(Ki=0.83 μM),正在开发中,用作针对 T 细胞的选择性免疫抑制剂。
Discription | CI 972 is a potent, orally active, and competitive inhibitor of purine nucleoside phosphorylase (PNP) (Ki=0.83 μM) under development as a T cell-selective immunosuppressive agent. |
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目录号 | A18598 |
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分子式 | C11H12ClN5OS |
分子量 | 297.76 |
CAS号 | 115787-68-3 |
SMILES | c1([nH]c2c(c(n1)=O)[nH]c(c2Cc1cscc1)N)N.Cl |
其他名称 | CI 972; CI972; CI-972. |
储存条件 | Store lyophilized at -20ºC, keep desiccated. |
Calculate the dilution required to prepare a stock solution. This equation is commonly abbreviated as: C1V1 = C2V2