CMPD-1
目录号: A16040
p38 MAPK 抑制剂
CMPD-1 是一种非 ATP 竞争性、选择性的 p38α介导的 MK2a(丝裂原活化蛋白激酶-2a)磷酸化抑制剂(表观 Ki = 330 nM)。
Discription | CMPD-1 is a non-ATP-competitive, selective inhibitor of p38α-mediated MK2a (mitogen-activated protein kinase-2a) phosphorylation (apparent Ki = 330 nM). | |||||
---|---|---|---|---|---|---|
Cell Research |
|
目录号 | A16040 |
---|---|
分子式 | C22H20FNO2 |
分子量 | 349.4 |
CAS号 | 41179-33-3 |
SMILES | FC1=CC=CC=C1C2=CC=C(C=C2)CCCC(NC(C=C3)=CC=C3O)=O |
其他名称 | CMPD1, CMPD 1 |
储存条件 | Store lyophilized at -20ºC, keep desiccated. |
Calculate the dilution required to prepare a stock solution. This equation is commonly abbreviated as: C1V1 = C2V2