Pelabresib (CPI 0610)
目录号: A16076
BET bromodomain 抑制剂
CPI 0610 是一种小分子抑制剂,针对 Bromodomain and Extra-Terminal (BET) 蛋白家族,具有潜在的抗肿瘤活性。
Discription | CPI 0610 is a small molecule inhibitor of the Bromodomain and Extra-Terminal (BET) family of proteins, with potential antineoplastic activity. | ||
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Targets |
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目录号 | A16076 |
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分子式 | C20H16ClN3O2 |
分子量 | 365.82 |
CAS号 | 1380087-89-7 |
SMILES | O=C(N)C[C@@H]1N=C(C2=CC=C(Cl)C=C2)C3=CC=CC=C3C4=C1ON=C4C |
其他名称 | CPI0610, CPI-0610 |
储存条件 | Store lyophilized at -20ºC, keep desiccated. |
In vitro | DMSO | 70 mg/mL (191.35 mM) | |
Water | Insoluble | ||
Ethanol | 12 mg/mL | ||
* <1 mg/ml means slightly soluble or insoluble. * Please note that Adooq tests the solubility of all compounds in-house, and the actual solubility may differ slightly from published values. This is normal and is due to slight batch-to-batch variations. |
Concentration / Solvent Volume / Mass | 1 mg | 5 mg | 10 mg |
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0.1 mM | 27.34 mL | 136.68 mL | 273.36 mL |
0.5 mM | 5.47 mL | 27.34 mL | 54.67 mL |
1 mM | 2.73 mL | 13.67 mL | 27.34 mL |
5 mM | 0.55 mL | 2.73 mL | 5.47 mL |
Calculate the dilution required to prepare a stock solution. This equation is commonly abbreviated as: C1V1 = C2V2