CPI-203

Name: CPI-203
SKU: A13068

目录号: A13068

BET bromodomain 抑制剂

Product Citations (1)

CPI-203 Chemical Structure

CAS NO. 1446144-04-2

CPI203是溴结构域和额外末端（BET）家族蛋白BRD4的新型有效，选择性和细胞渗透性抑制剂，IC50为?37 nM（BRD4α筛选试验）。

库存：现货

规格	价格	数量
5 mg	￥ 630.00
10 mg	￥ 1,190.00
25 mg	￥ 2,450.00
50 mg	￥ 3,850.00

大包装询价

或

添加到收藏

产品仅用于科学研究，不针对患者销售，望谅解.

产品详情

生物活性

CPI203是溴结构域和额外末端（BET）家族蛋白BRD4的新型有效，选择性和细胞渗透性抑制剂，IC50为?37 nM（BRD4α筛选试验）。

溶解度 *

In vitro	DMSO	Warmed: 78 mg/mL (195.04 mM)
	Water	Insoluble
	Ethanol	5 mg/mL (12.5 mM)
* <1 mg/ml means slightly soluble or insoluble. * Please note that Adooq tests the solubility of all compounds in-house, and the actual solubility may differ slightly from published values. This is normal and is due to slight batch-to-batch variations.

制备储备液

Concentration / Solvent Volume / Mass	1 mg	5 mg	10 mg
0.1 mM	25.01 mL	125.03 mL	250.06 mL
0.5 mM	5 mL	25.01 mL	50.01 mL
1 mM	2.5 mL	12.5 mL	25.01 mL
5 mM	0.5 mL	2.5 mL	5 mL

*The above data is based on the productmolecular weight 399.9. Batch specific molecular weights may vary from batch to batch due to solvent of hydration, which will affect the solvent volumes required to prepare stock solutions.

化学数据

目录号	A13068
作用机制	Inhibitor (抑制剂)
M. Wt	399.9
Formula	C19H18ClN5OS
Purity	>99%
Storage	Store lyophilized at -20ºC, keep desiccated. In lyophilized form, the chemical is stable for 36 months. In solution, store at -20ºC and use within 3 months to prevent loss of potency. Aliquot to avoid multiple freeze/thaw cycles.
CAS No.	1446144-04-2
Synonyms	0
SMILES	CC1=C(SC2=C1C(=N[C@H](C3=NN=C(N32)C)CC(=O)N)C4=CC=C(C=C4)Cl)C