CRT-0066101
目录号: A16318
PKD 抑制剂
CRT-0066101 是一种强效的 蛋白激酶D (PKD) 抑制剂;它能抑制所有 PKD 同型体(IC50 值分别为 PKD1、PKD3 和 PKD2 的 1、2 和 2.5 nM)。
Discription | CRT-0066101, potent inhibitor of protein kinase D (PKD); inhibits all PKD isoforms (IC50 values are 1, 2 and 2.5 nM for PKD1, PKD3 and PKD2 respectively). | ||
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Targets |
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目录号 | A16318 |
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分子式 | C18H22N6O.2HCl |
分子量 | 411.33 |
CAS号 | 1883545-60-5 |
SMILES | Cl.Cl.Cn1cc(cn1)c3cc(c2nc(NC[C@H](N)CC)ccn2)c(O)cc3 |
其他名称 | CRT 0066101, CRT0066101 |
储存条件 | Store lyophilized at -20ºC, keep desiccated. |
In vitro | DMSO | Warmed: 25 mg/mL (60.77 mM) | |
Water | 80 mg/mL (194.49 mM) | ||
Ethanol | Warmed: 2 mg/mL | ||
* <1 mg/ml means slightly soluble or insoluble. * Please note that Adooq tests the solubility of all compounds in-house, and the actual solubility may differ slightly from published values. This is normal and is due to slight batch-to-batch variations. |
Concentration / Solvent Volume / Mass | 1 mg | 5 mg | 10 mg |
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0.1 mM | 24.31 mL | 121.56 mL | 243.11 mL |
0.5 mM | 4.86 mL | 24.31 mL | 48.62 mL |
1 mM | 2.43 mL | 12.16 mL | 24.31 mL |
5 mM | 0.49 mL | 2.43 mL | 4.86 mL |
Calculate the dilution required to prepare a stock solution. This equation is commonly abbreviated as: C1V1 = C2V2