CX-4945 sodium salt
目录号: A16234
CK2 抑制剂
CX-4945 钠盐是一种强效且选择性的 ATP-竞争性小分子蛋白激酶 CK2 抑制剂,其对重组人类 CK2α 的 Ki 和 IC50 分别为 0.38 nM 和 1 nM。
Discription | CX-4945 sodium salt is a potent and selective ATP-competitive small molecule protein kinase CK2 inhibitor with a Ki and an IC50 of 0.38 and 1 nM for recombinant human CK2α, respectively. | ||
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Targets |
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目录号 | A16234 |
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分子式 | C19H11ClN3NaO2 |
分子量 | 371.75 |
CAS号 | 1309357-15-0 |
SMILES | C1=CC(=CC(=C1)Cl)NC2=NC3=C(C=CC(=C3)C(=O)[O-])C4=C2C=CN=C4.[Na+] |
其他名称 | Silmitasertib sodium salt |
储存条件 | Store lyophilized at -20ºC, keep desiccated. |
In vitro | DMSO | 65 mg/mL (174.84 mM) | |
Water | 65 mg/mL (174.84 mM) | ||
Ethanol | Insoluble | ||
* <1 mg/ml means slightly soluble or insoluble. * Please note that Adooq tests the solubility of all compounds in-house, and the actual solubility may differ slightly from published values. This is normal and is due to slight batch-to-batch variations. |
Concentration / Solvent Volume / Mass | 1 mg | 5 mg | 10 mg |
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0.1 mM | 26.9 mL | 134.5 mL | 269 mL |
0.5 mM | 5.38 mL | 26.9 mL | 53.8 mL |
1 mM | 2.69 mL | 13.45 mL | 26.9 mL |
5 mM | 0.54 mL | 2.69 mL | 5.38 mL |
Calculate the dilution required to prepare a stock solution. This equation is commonly abbreviated as: C1V1 = C2V2