CX-6258 hydrochloride hydrate
目录号: A15055
Pim 抑制剂
CX-6258 hydrochloride hydrate 是一种效力强大的口服 Pim 1/2/3 kinase 抑制剂(IC50=5 nM/25 nM/16 nM),具有出色的生化效力和激酶选择性。
Discription | CX-6258 hydrochloride hydrate is a potent, orally efficacious Pim 1/2/3 kinase(IC50=5 nM/25 nM/16 nM) inhibitor with excellent biochemical potency and kinase selectivity. |
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目录号 | A15055 |
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分子式 | C26H27Cl2N3O4 |
分子量 | 516.42 |
CAS号 | 1353858-99-7 |
SMILES | CN1CCCN(CC1)C(=O)C2=CC=CC(=C2)C3=CC=C(O3)C=C4C5=C(C=CC(=C5)Cl)NC4=O.O.Cl |
其他名称 | CX6258 hydrochloride hydrate, CX 6258 hydrochloride hydrate |
储存条件 | Store lyophilized at -20ºC, keep desiccated. |
Calculate the dilution required to prepare a stock solution. This equation is commonly abbreviated as: C1V1 = C2V2