DBPR108
目录号: A21833
DPP4 抑制剂
DBPR108 是一种高效、选择性且可口服生物利用的二肽衍生的 DPP4 抑制剂,其 IC50 为 15 nM;对 DDP8 和 DPP9 无抑制作用。
Discription | DBPR108 is a potent, selective, and orally bioavailable dipeptide-derived inhibitor of DPP4 with IC50 of 15 nM; no inhibition on DDP8 and DPP9. |
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目录号 | A21833 |
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分子式 | C16H25FN4O2 |
分子量 | 324.39 |
CAS号 | 1186426-66-3 |
SMILES | N#C[C@H]1N(C(CNC(C)(C)CC(N2CCCC2)=O)=O)C[C@@H](F)C1 |
其他名称 | DBPR 108, DBPR 108 |
储存条件 | Store lyophilized at -20ºC, keep desiccated. |
Calculate the dilution required to prepare a stock solution. This equation is commonly abbreviated as: C1V1 = C2V2